Dehydrogenase
Metabolic Enzyme/Protease
11β-HSD(15)
15-PGDH(1)
ACC(10)
ACE(15)
AChE(47)
Adenylate Cyclase(12)
ALDH(14)
Aldose Reductase(5)
Aminopeptidase(19)
BACE(19)
Casein Kinase(51)
CAT(5)
Cathepsin(9)
CETP(13)
COMT(2)
CPG2(1)
CYPs(6)
Decarboxylase(3)
Dehydrogenase(131)
DGAT(4)
Dopamine beta-hydroxylase(2)
DPP(32)
Elastase(6)
FAAH(28)
Factor Xa(31)
Fatty Acid Synthase(17)
Ftase(2)
FXR(26)
Glucokinase(1)
GSNOR(2)
Guanylate Cyclase(13)
HMGCR(17)
IDH(7)
IDO(20)
IMPDH(2)
LDH(2)
LDL(8)
Lipase(17)
Lipid(12)
MAGL(6)
MAO(72)
MMP(78)
NAMPT(12)
Neprilysin(7)
Other Targets(10)
P450(112)
PAI-1(9)
Phosphatase(95)
Phospholipase(65)
PPAR(115)
Protein Phosphatase/PTP(6)
Renin(8)
Retinoid Receptor(37)
SCD(6)
Steroid Sulfatase (STS)(2)
Thioredoxin(1)
TPH(5)
Transferase(37)
Vitamin(44)
Xanthine Oxidase (XAO)(11)
Dehydrogenase
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(E/Z)-Ginkgolic acid C17:2
产品货号 : M37748
cas no: 102811-39-2
(E/Z)-Ginkgolic acid C17:2 来自银杏,可靶向人二氢乳清酸脱氢酶 (DHODH). -
SW209049
产品货号 : M37687
cas no: 1673558-59-2
SW209049 is a stearoyl-CoA 9-desaturase inhibitor. SW209049 exhivits potent activity against H2122 cell with IC50 of 0.13uM. -
G6PDi-1 B
产品货号 : M37586
cas no: 2457232-14-1
G6PDi-1 是一种可逆的非竞争性6-磷酸葡萄糖脱氢酶 (G6PD) 抑制剂,对人 G6PD IC50 为 0.07 μM。G6PDi-1 最强烈地消耗淋巴细胞中的 NADPH。G6PDi-1 显着降低 T 细胞中炎性细胞因子的产生。 -
IDH2R140Q-IN-2
产品货号 : M37247
cas no: 2749568-16-7
IDH2R140Q-IN-2 (化合物 36) 是一种具有口服活性的 IDH2R140Q 抑制剂 (IC50: 29 nM)。IDH2R140Q-IN-2 减少表达突变 IDH2R140Q 的 TF-1 细胞系中 D2HG 的产生 (IC50: 10 nM)。IDH2R140Q-IN-2 抑制肿瘤组织中的 D2HG 水平。IDH2R140Q-IN-2 可用于急性髓系白血病 (AML) 的研究。 -
WAY-311610
产品货号 : M36983
cas no: 314051-55-3
WAY-311610 is an 11β-hydroxysteroid dehydrogenase HSD11B1 inhibitor that inhibits the 11β-HSD1 enzyme with an IC = 0.34 μM.It can be used to study neuropathic pain, inflammatory pain, and occipital neuralgia.