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Dimethylenastron
CAS No. 863774-58-7
Dimethylenastron ( Dimethylenastron )
产品货号. M16256 CAS No. 863774-58-7
A small molecule inhibitor of the mitotic kinesin Eg5; inhibits endothelial cell proliferation and migration in vitro.
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| 规格 | 价格/人民币 | 库存 | 数量 |
| 2MG | ￥348 | 有现货 |
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| 5MG | ￥543 | 有现货 |
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| 10MG | ￥721 | 有现货 |
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| 25MG | ￥1418 | 有现货 |
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| 50MG | ￥2657 | 有现货 |
|
| 100MG | ￥4301 | 有现货 |
|
| 200MG | 获取报价 | 有现货 |
|
| 500MG | 获取报价 | 有现货 |
|
| 1G | 获取报价 | 有现货 |
|
生物学信息
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产品名称Dimethylenastron
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注意事项本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
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产品简述A small molecule inhibitor of the mitotic kinesin Eg5; inhibits endothelial cell proliferation and migration in vitro.
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产品描述A small molecule inhibitor of the mitotic kinesin Eg5; inhibits endothelial cell proliferation and migration in vitro; exhibits a shorter mitotic arrest, bipolar or multipolar karyokinesis, followed by apoptosis of the daughter cells in dimethylenastron-treated tetraploid cells.
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同义词Dimethylenastron
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通路Cytoskeleton/Cell Adhesion Molecules
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靶点Kinesin
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受体Eg5
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研究领域Cancer
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适应症——
化学信息
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CAS Number863774-58-7
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分子量302.39
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分子式C16H18N2O2S
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纯度>98% (HPLC)
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溶解度DMSO: ≥ 31 mg/mL
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SMILESO=C1C2=C(NC(NC2C3=CC=CC(O)=C3)=S)CC(C)(C)C1
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化学全称5(1H)-Quinazolinone, 2,3,4,6,7,8-hexahydro-4-(3-hydroxyphenyl)-7,7-dimethyl-2-thioxo-
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1. Rello-Varona S, et al. Cell Cycle. 2009 Apr 1;8(7):1030-5.
2. Exertier P, et al. Oncotarget. 2013 Dec;4(12):2302-16.
3. Kaan HY, et al. J Med Chem. 2010 Aug 12;53(15):5676-83.
2. Exertier P, et al. Oncotarget. 2013 Dec;4(12):2302-16.
3. Kaan HY, et al. J Med Chem. 2010 Aug 12;53(15):5676-83.
产品手册
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