Tebanicline
CAS No. 198283-73-7
Tebanicline ( —— )
产品货号. M17413 CAS No. 198283-73-7
Tebanicline (ABT-594, Ebanicline) acts as a partial agonist at neuronal nicotinic acetylcholine receptors, binding to both the α3β4 and the α4β2 subtypes.
纯度: 98%
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
规格 | 价格/人民币 | 库存 | 数量 |
2MG | ¥450 | 有现货 |
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5MG | ¥811 | 有现货 |
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10MG | ¥1270 | 有现货 |
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25MG | ¥2655 | 有现货 |
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50MG | ¥3643 | 有现货 |
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100MG | 获取报价 | 有现货 |
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200MG | 获取报价 | 有现货 |
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500MG | 获取报价 | 有现货 |
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1G | 获取报价 | 有现货 |
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生物学信息
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产品名称Tebanicline
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注意事项本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
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产品简述Tebanicline (ABT-594, Ebanicline) acts as a partial agonist at neuronal nicotinic acetylcholine receptors, binding to both the α3β4 and the α4β2 subtypes.
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产品描述Tebanicline (ABT-594, Ebanicline) acts as a partial agonist at neuronal nicotinic acetylcholine receptors, binding to both the α3β4 and the α4β2 subtypes. Tebanicline is an effective synthetic nicotinic (non-opioid) analgesic drug developed by Abbott. It was developed as a less toxic analog of the potent poison dart frog-derived compound epibatidine, which is some 200x stronger than morphine as an analgesic but produces extremely dangerous toxic side effects. Like epibatidine, Tebanicline showed potent analgesic activity against neuropathic pain in both animal and human trials, but with far less toxicity than its parent compound.
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同义词——
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通路Cell Cycle/DNA Damage
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靶点PLK
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受体nAChR
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研究领域——
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适应症——
化学信息
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CAS Number198283-73-7
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分子量198.65
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分子式C9H11ClN2O
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纯度98%
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溶解度——
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SMILESC1CN[C@H]1COc1cnc(cc1)Cl
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化学全称——
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1. Hayashi T, et al.Neurosci Lett. 2016 Dec 7;638:46-50.
产品手册
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