Rigosertib
CAS No. 1225497-78-8
Rigosertib ( ON-01910 )
产品货号. M10864 CAS No. 1225497-78-8
Rigosertib (ON-01910) is a non-ATP-competitive inhibitor of PLK1 with IC50 of 9 nM.
纯度: >98%(HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
规格 | 价格/人民币 | 库存 | 数量 |
2MG | ¥275 | 有现货 |
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5MG | ¥446 | 有现货 |
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10MG | ¥786 | 有现货 |
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25MG | ¥1563 | 有现货 |
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50MG | ¥2940 | 有现货 |
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100MG | ¥5038 | 有现货 |
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200MG | 获取报价 | 有现货 |
|
500MG | 获取报价 | 有现货 |
|
1G | 获取报价 | 有现货 |
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生物学信息
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产品名称Rigosertib
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注意事项本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
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产品简述Rigosertib (ON-01910) is a non-ATP-competitive inhibitor of PLK1 with IC50 of 9 nM.
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产品描述Rigosertib (ON-01910) is a non-ATP-competitive inhibitor of PLK1 with IC50 of 9 nM. It shows 30-fold greater selectivity against Plk2 and no activity to Plk3. Phase 3.
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同义词ON-01910
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通路Cell Cycle/DNA Damage
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靶点PLK
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受体PLK1
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研究领域Cancer
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适应症——
化学信息
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CAS Number1225497-78-8
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分子量473.47
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分子式C21H24NNaO8S
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纯度>98%(HPLC)
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溶解度Water: 95 mg/mL (200.64 mM); DMSO: 95 mg/mL (200.64 mM)
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SMILESCOC1=C(C=C(C=C1)CS(=O)(=O)/C=C/C2=C(C=C(C=C2OC)OC)OC)NCC(=O)[O-].[Na+]
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化学全称——
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1.Gumireddy K, et al. Y Cell, 2005, 7(3), 275-286.
产品手册
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