Poloxin
CAS No. 321688-88-4
Poloxin ( —— )
产品货号. M24255 CAS No. 321688-88-4
Poloxin is a non-ATP competitive Polo-like Kinase 1 inhibitor. It targets the polo-box domain (IC50: appr 4.8 μM).
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
规格 | 价格/人民币 | 库存 | 数量 |
10MG | ¥389 | 有现货 |
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25MG | ¥932 | 有现货 |
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50MG | ¥1669 | 有现货 |
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100MG | ¥2479 | 有现货 |
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200MG | ¥3694 | 有现货 |
|
500MG | 获取报价 | 有现货 |
|
1G | 获取报价 | 有现货 |
|
生物学信息
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产品名称Poloxin
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注意事项本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
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产品简述Poloxin is a non-ATP competitive Polo-like Kinase 1 inhibitor. It targets the polo-box domain (IC50: appr 4.8 μM).
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产品描述Poloxin is a non-ATP competitive Polo-like Kinase 1 inhibitor. It targets the polo-box domain (IC50: appr 4.8 μM).
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同义词——
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通路Cell Cycle/DNA Damage
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靶点PLK
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受体PLK1;PLK2;PLK3
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研究领域——
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适应症——
化学信息
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CAS Number321688-88-4
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分子量297.4
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分子式C18H19NO3
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纯度>98% (HPLC)
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溶解度DMSO:14 mg/mL (43.72 mM; Need ultrasonic)
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SMILESCC(C)C(C(C=C1C)=O)=C/C1=N/OC(c1c(C)cccc1)=O
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化学全称——
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1.Yuan J, et al. Polo-box domain inhibitor poloxin activates the spindle assembly checkpoint and inhibits tumor growth in vivo. Am J Pathol. 2011 Oct;179(4):2091-9.
产品手册
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