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TAS-115
CAS No. 1190836-34-0
TAS-115 ( H2OL3Q4XRD; 4-(2-Fluoro-4-(3-(2-phenylacetyl)thioureido)phenoxy)-7-methoxy-N-methylquinoline-6-carboxamide; pamufetinib )
产品货号. M23360 CAS No. 1190836-34-0
TAS-115 is a potent inhibitor of VEGFR and hepatocyte growth factor receptor (c-Met/HGFR)-targeted kinase(IC50s of 30 and 32 nM for rVEGFR2 and rMET, respectively).
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| 规格 | 价格/人民币 | 库存 | 数量 |
| 5MG | ￥1458 | 有现货 |
|
| 10MG | ￥2155 | 有现货 |
|
| 25MG | ￥3653 | 有现货 |
|
| 50MG | ￥5370 | 有现货 |
|
| 100MG | ￥7655 | 有现货 |
|
| 200MG | 获取报价 | 有现货 |
|
| 500MG | 获取报价 | 有现货 |
|
| 1G | 获取报价 | 有现货 |
|
生物学信息
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产品名称TAS-115
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注意事项本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
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产品简述TAS-115 is a potent inhibitor of VEGFR and hepatocyte growth factor receptor (c-Met/HGFR)-targeted kinase(IC50s of 30 and 32 nM for rVEGFR2 and rMET, respectively).
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产品描述TAS-115 is a potent inhibitor of VEGFR and hepatocyte growth factor receptor (c-Met/HGFR)-targeted kinase(IC50s of 30 and 32 nM for rVEGFR2 and rMET, respectively).
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同义词H2OL3Q4XRD; 4-(2-Fluoro-4-(3-(2-phenylacetyl)thioureido)phenoxy)-7-methoxy-N-methylquinoline-6-carboxamide; pamufetinib
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通路Angiogenesis
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靶点VEGFR
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受体VEGFR2;c-Met
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研究领域——
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适应症——
化学信息
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CAS Number1190836-34-0
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分子量518.6
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分子式C27H23FN4O4S
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纯度>98% (HPLC)
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溶解度——
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SMILESCNC(c(cc1c(Oc(ccc(NC(NC(Cc2ccccc2)=O)=S)c2)c2F)ccnc1c1)c1OC)=O
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化学全称——
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1.Fujita H, et al. The novel VEGF receptor/MET-targeted kinase inhibitor TAS-115 has marked in vivo antitumor properties and a favorable tolerability profile. Mol Cancer Ther. 2013 Dec;12(12):2685-96.
产品手册
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