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TAK-593
CAS No. 1005780-62-0
TAK-593 ( —— )
产品货号. M23210 CAS No. 1005780-62-0
TAK-593 is an effective VEGFR and PDGFR family inhibitor.
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| 规格 | 价格/人民币 | 库存 | 数量 |
| 5MG | ￥794 | 有现货 |
|
| 10MG | ￥1393 | 有现货 |
|
| 25MG | ￥2746 | 有现货 |
|
| 50MG | ￥4253 | 有现货 |
|
| 100MG | ￥6148 | 有现货 |
|
| 200MG | 获取报价 | 有现货 |
|
| 500MG | 获取报价 | 有现货 |
|
| 1G | 获取报价 | 有现货 |
|
生物学信息
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产品名称TAK-593
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注意事项本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
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产品简述TAK-593 is an effective VEGFR and PDGFR family inhibitor.
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产品描述TAK-593 is an effective VEGFR and PDGFR family inhibitor (IC50s: 3.2, 0.95, 1.1, 4.3, and 13 nM for VEGFR1, VEGFR2, VEGFR3, PDFGRα, and PDFGRβ, respectively).
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同义词——
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通路Angiogenesis
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靶点VEGFR
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受体VEGFR1;VEGFR2;VEGFR3;PDGFRα;PDGFRβ;PDGFRαV561D
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研究领域——
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适应症——
化学信息
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CAS Number1005780-62-0
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分子量445.5
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分子式C23H23N7O3
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纯度>98% (HPLC)
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溶解度DMSO:45 mg/mL (101.02 mM)
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SMILESO=C(C1=CC(C)=NN1C)NC2=CC(OC3=NN4C(C=C3)=NC(NC(C5CC5)=O)=C4)=CC=C2C
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化学全称——
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1.Miyamoto N, et al. Discovery of N-[5-({2-[(cyclopropylcarbonyl)amino]imidazo[1,2-b]pyridazin-6-yl}oxy)-2-methylphenyl]-1,3-dimethyl-1H-pyrazole-5-carboxamide (TAK-593), a highly potent VEGFR2 kinase inhibitor. Bioorg Med Chem. 2013 Apr 15;21(8):2333-2345.
产品手册
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