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Olinone
CAS No. 1770789-37-1
Olinone ( Olinone )
产品货号. M12666 CAS No. 1770789-37-1
Olinone is a selective inhibitor for the BET BRD1 with Kd of 3.4/3.7/8.6 uM for BRD4-BrD1/BRD3-BrD1/BRD2-BrD1, respectively.
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| 规格 | 价格/人民币 | 库存 | 数量 |
| 5MG | ￥7857 | 有现货 |
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| 50MG | ￥16038 | 有现货 |
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| 100MG | ￥20250 | 有现货 |
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| 200MG | 获取报价 | 有现货 |
|
| 500MG | 获取报价 | 有现货 |
|
| 1G | 获取报价 | 有现货 |
|
生物学信息
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产品名称Olinone
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注意事项本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
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产品简述Olinone is a selective inhibitor for the BET BRD1 with Kd of 3.4/3.7/8.6 uM for BRD4-BrD1/BRD3-BrD1/BRD2-BrD1, respectively.
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产品描述Olinone is a selective inhibitor for the BET BRD1 with Kd of 3.4/3.7/8.6 uM for BRD4-BrD1/BRD3-BrD1/BRD2-BrD1, respectively, shows high selectivity over BET BRD2 (Kd>300 uM); accelerates the progression of mouse primary oligodendrocyte progenitors toward differentiation.
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同义词Olinone
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通路Chromatin/Epigenetic
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靶点Bromodomain
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受体Bromodomain
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研究领域——
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适应症——
化学信息
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CAS Number1770789-37-1
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分子量299.37
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分子式C17H21N3O2
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纯度>98% (HPLC)
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溶解度——
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SMILESCC(NCCCCN1C(CCN2)=C(C2=O)C3=C1C=CC=C3)=O
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化学全称N-[4-(1-Oxo-1,2,3,4-tetrahydro-pyrido[4,3-b]indol-5-yl)-butyl]-acetamide
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1. Gacias M, et al. Chem Biol. 2014 Jul 17;21(7):841-54.
2. Chiang CM. Chem Biol. 2014 Jul 17;21(7):804-6.
3. Zhao L, et J Neuroinflammation. 2017 Jan 19;14(1):14.al.
2. Chiang CM. Chem Biol. 2014 Jul 17;21(7):804-6.
3. Zhao L, et J Neuroinflammation. 2017 Jan 19;14(1):14.al.
产品手册
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