BETi-211 ( BETi 211;BETi211 )

产品货号. M13114 CAS No. 1995867-02-1

COA

Datasheet

HNMR

HPLC

MSDS

Handing Instructions

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产品名称

BETi-211
注意事项

本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
产品简述

A novel potent small-molecule BET bromodomain (BRD) inhibitor that binds to BET proteins with Ki values of <1 nM.
产品描述

A novel potent small-molecule BET bromodomain (BRD) inhibitor that binds to BET proteins with Ki values of <1 nM; exhibits >10-100 times more potent than RX-37, JQ-1, OTX-015 or IBET-762.
同义词

BETi 211;BETi211
通路

Chromatin/Epigenetic
靶点

Bromodomain
受体

Bromodomain
研究领域

——
适应症

——

CAS Number

1995867-02-1
分子量

487.56
分子式

C26H29N7O3
纯度

>98% (HPLC)
溶解度

——
SMILES

COCC1=NC(NC2=CC(C3CC3)=NN2CC)=C4C(NC5=C4C=C(OC)C(C6=C(C)ON=C6C)=C5)=N1
化学全称

N-(3-cyclopropyl-1-ethyl-1H-pyrazol-5-yl)-7-(3,5-dimethylisoxazol-4-yl)-6-methoxy-2-(methoxymethyl)-9H-pyrimido[4,5-b]indol-4-amine

计算器

产品手册

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