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LY2119620

CAS No. 886047-22-9

LY2119620 ( LY2119620; LY 2119620; LY-2119620 )

产品货号. M17642 CAS No. 886047-22-9

LY2119620 is a specific, and allosteric agonist of human M2 and M4 muscarinic acetylcholine receptors.

纯度: 98%

COA Datasheet HNMR HPLC MSDS Handing Instructions
规格 价格/人民币 库存 数量
2MG ¥591 有现货
5MG ¥1013 有现货
10MG ¥1604 有现货
25MG ¥3094 有现货
50MG ¥4609 有现货
100MG ¥6634 有现货
200MG 获取报价 有现货
500MG 获取报价 有现货
1G 获取报价 有现货

生物学信息

  • 产品名称
    LY2119620
  • 注意事项
    本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
  • 产品简述
    LY2119620 is a specific, and allosteric agonist of human M2 and M4 muscarinic acetylcholine receptors.
  • 产品描述
    LY2119620 is a positive allosteric modulator of the M2 and M4 muscarinic acetylcholine receptors (mAChRs).
  • 同义词
    LY2119620; LY 2119620; LY-2119620
  • 通路
    Others
  • 靶点
    Other Targets
  • 受体
    M2 mAChR;M4 mAChR
  • 研究领域
    Neurological Disease
  • 适应症
    ——

化学信息

  • CAS Number
    886047-22-9
  • 分子量
    437.94
  • 分子式
    C19H24ClN5O3S
  • 纯度
    98%
  • 溶解度
    DMSO : 67.5 mg/mL. 154.13 mM; H2O : < 0.1 mg/mL
  • SMILES
    CN1CCN(CC1)C(=O)COc1nc2sc(C(=O)NC3CC3)c(N)c2c(C)c1Cl
  • 化学全称
    3-amino-5-chloro-N-cyclopropyl-4-methyl-6-[2-(4-methyl-1-piperazinyl)-2-oxoethoxy]-thieno[2,3-b]pyridine-2-carboxamide

运输与储存

  • 储存条件
    (-20℃)
  • 运输条件
    With Ice Pack
  • 稳定性
    ≥ 2 years

参考文献

1.Croy C H, Schober D A, Xiao H, et al. Characterization of the novel positive allosteric modulator, LY2119620, at the muscarinic M(2) and M(4) receptors.[J]. Molecular Pharmacology, 2014, 86(1):106-115.
产品手册
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