LY2119620
CAS No. 886047-22-9
LY2119620 ( LY2119620; LY 2119620; LY-2119620 )
产品货号. M17642 CAS No. 886047-22-9
LY2119620 is a specific, and allosteric agonist of human M2 and M4 muscarinic acetylcholine receptors.
纯度: 98%
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
规格 | 价格/人民币 | 库存 | 数量 |
2MG | ¥591 | 有现货 |
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5MG | ¥1013 | 有现货 |
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10MG | ¥1604 | 有现货 |
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25MG | ¥3094 | 有现货 |
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50MG | ¥4609 | 有现货 |
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100MG | ¥6634 | 有现货 |
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200MG | 获取报价 | 有现货 |
|
500MG | 获取报价 | 有现货 |
|
1G | 获取报价 | 有现货 |
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生物学信息
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产品名称LY2119620
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注意事项本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
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产品简述LY2119620 is a specific, and allosteric agonist of human M2 and M4 muscarinic acetylcholine receptors.
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产品描述LY2119620 is a positive allosteric modulator of the M2 and M4 muscarinic acetylcholine receptors (mAChRs).
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同义词LY2119620; LY 2119620; LY-2119620
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通路Others
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靶点Other Targets
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受体M2 mAChR;M4 mAChR
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研究领域Neurological Disease
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适应症——
化学信息
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CAS Number886047-22-9
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分子量437.94
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分子式C19H24ClN5O3S
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纯度98%
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溶解度DMSO : 67.5 mg/mL. 154.13 mM; H2O : < 0.1 mg/mL
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SMILESCN1CCN(CC1)C(=O)COc1nc2sc(C(=O)NC3CC3)c(N)c2c(C)c1Cl
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化学全称3-amino-5-chloro-N-cyclopropyl-4-methyl-6-[2-(4-methyl-1-piperazinyl)-2-oxoethoxy]-thieno[2,3-b]pyridine-2-carboxamide
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1.Croy C H, Schober D A, Xiao H, et al. Characterization of the novel positive allosteric modulator, LY2119620, at the muscarinic M(2) and M(4) receptors.[J]. Molecular Pharmacology, 2014, 86(1):106-115.
产品手册
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