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PSB-603
CAS No. 1092351-10-4
PSB-603 ( PSB 603 )
产品货号. M27690 CAS No. 1092351-10-4
Adenosine A2B receptor antagonist.
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| 规格 | 价格/人民币 | 库存 | 数量 |
| 5MG | ￥3224 | 有现货 |
|
| 10MG | ￥4795 | 有现货 |
|
| 25MG | ￥7671 | 有现货 |
|
| 50MG | ￥10368 | 有现货 |
|
| 100MG | ￥14013 | 有现货 |
|
| 200MG | 获取报价 | 有现货 |
|
| 500MG | 获取报价 | 有现货 |
|
| 1G | 获取报价 | 有现货 |
|
生物学信息
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产品名称PSB-603
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注意事项本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
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产品简述Adenosine A2B receptor antagonist.
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产品描述Adenosine A2B receptor antagonist.(In Vitro):In peripheral T cells, PSB-603 (100 nM) inhibits NECA-stimulated IL-6 release about 3-fold. PSB-603 (10 μM) shows no affinity for the human and rat A1 and A2A and human A3 receptors.(In Vivo):PSB-603 (5 mg/kg; i.p.) significantly reduces inflammation in local and systemic mice models of inflammation. In the inflamed paw, PSB-603 significantly decreases the levels of the inflammatory cytokines including IL-6, TNF-α and of ROS. PSB-603 reduces inflammation of the peritoneum by decreasing the infiltration of leukocytes.
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同义词PSB 603
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通路Others
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靶点Other Targets
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受体——
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研究领域——
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适应症——
化学信息
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CAS Number1092351-10-4
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分子量529.0
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分子式C24H25ClN6O4S
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纯度>98% (HPLC)
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溶解度——
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SMILESCCCn1c(O)nc2nc([nH]c2c1=O)-c1ccc(cc1)S(=O)(=O)N1CCN(CC1)c1ccc(Cl)cc1
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化学全称——
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1.Edward Scolnick, et al. Uses of paralog-selective inhibitors of gsk3 kinases. US20160375006A1.
产品手册
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