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LDN212854
CAS No. 1432597-26-6
LDN212854 ( LDN212854; LDN 212854; LDN-212854 )
产品货号. M11840 CAS No. 1432597-26-6
LDN-212854 is a novel BMP inhibitor that exhibits substantially greater selectivity for BMP versus the TGF-β type I receptors.
纯度: >98%(HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| 规格 | 价格/人民币 | 库存 | 数量 |
| 5MG | ￥794 | 有现货 |
|
| 10MG | ￥1499 | 有现货 |
|
| 25MG | ￥3013 | 有现货 |
|
| 50MG | ￥4504 | 有现货 |
|
| 100MG | ￥6342 | 有现货 |
|
| 200MG | 获取报价 | 有现货 |
|
| 500MG | 获取报价 | 有现货 |
|
| 1G | 获取报价 | 有现货 |
|
生物学信息
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产品名称LDN212854
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注意事项本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
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产品简述LDN-212854 is a novel BMP inhibitor that exhibits substantially greater selectivity for BMP versus the TGF-β type I receptors.
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产品描述LDN-212854 is a novel BMP inhibitor that exhibits substantially greater selectivity for BMP versus the TGF-β type I receptors; possesses a bias towards ALK2(IC50=1.3 nM) versus ALK1 and ALK3 compared to other inhibitors.
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同义词LDN212854; LDN 212854; LDN-212854
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通路Angiogenesis
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靶点ALK
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受体ALK1; ALK2; ALK3; ALK4; ALK5
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研究领域Cancer
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适应症——
化学信息
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CAS Number1432597-26-6
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分子量406.48
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分子式C25H22N6
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纯度>98%(HPLC)
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溶解度DMSO: 81 mg/mL warmed (199.27 mM)
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SMILESC12=C(C3=C4N=CC(C5=CC=C(N6CCNCC6)C=C5)=CN4N=C3)C=CC=C1N=CC=C2
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化学全称5-(6-(4-(piperazin-1-yl)phenyl)pyrazolo[1,5-a]pyrimidin-3-yl)quinoline
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
产品手册
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