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AP26113
CAS No. 1197958-12-5
AP26113 ( —— )
产品货号. M10707 CAS No. 1197958-12-5
AP26113 is a potent ALK inhibitor with IC50 of 0.62 nM in a cell-free assay.
纯度: >98%(HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| 规格 | 价格/人民币 | 库存 | 数量 |
| 2MG | ￥243 | 有现货 |
|
| 5MG | ￥381 | 有现货 |
|
| 10MG | ￥543 | 有现货 |
|
| 25MG | ￥786 | 有现货 |
|
| 50MG | ￥1191 | 有现货 |
|
| 100MG | ￥2001 | 有现货 |
|
| 200MG | ￥2981 | 有现货 |
|
| 500MG | ￥4828 | 有现货 |
|
| 1G | 获取报价 | 有现货 |
|
生物学信息
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产品名称AP26113
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注意事项本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
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产品简述AP26113 is a potent ALK inhibitor with IC50 of 0.62 nM in a cell-free assay.
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产品描述AP26113 is a potent ALK inhibitor with IC50 of 0.62 nM in a cell-free assay, demonstrated ability overcome Crizotinib resistance mediated by a L1196M mutation. Phase 2.
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同义词——
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通路Angiogenesis
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靶点ALK
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受体ALK; EGFR (C797S/del19); EGFR (del19); EGFR (del19); IGF-1R
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研究领域Cancer
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适应症——
化学信息
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CAS Number1197958-12-5
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分子量529.01
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分子式C26H34ClN6O2P
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纯度>98%(HPLC)
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溶解度Ethanol: 106 mg/mL (200.37 mM); DMSO: 45 mg/mL (85.06 mM)
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SMILESCOC1=C(NC2=NC=C(Cl)C(NC3=CC=CC=C3P(C)(C)=O)=N2)C=CC(=C1)N1CCC(CC1)N(C)C
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化学全称——
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1.Sen Zhang, et al. Y Research: April 15, 2010; Volume 70, Issue 8, Supplement 1
产品手册
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