GSK-1
CAS No. 912953-25-4
GSK-1 ( —— )
产品货号. M16555 CAS No. 912953-25-4
GSK-1 is an ATP-competitive inhibitor of the mitotic kinesin KSP with HCT116 cell IC50 of 36 nM.
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
规格 | 价格/人民币 | 库存 | 数量 |
100MG | 获取报价 | 有现货 |
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200MG | 获取报价 | 有现货 |
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500MG | 获取报价 | 有现货 |
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1G | 获取报价 | 有现货 |
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生物学信息
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产品名称GSK-1
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注意事项本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
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产品简述GSK-1 is an ATP-competitive inhibitor of the mitotic kinesin KSP with HCT116 cell IC50 of 36 nM.
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产品描述GSK-1 is an ATP-competitive inhibitor of the mitotic kinesin KSP with HCT116 cell IC50 of 36 nM; induces monopolar spindle formation in SKOV3 cells, and shows markedly greater potency (IC50 of 0.5 nM) in the ispinesib-resistant HCT116-D130V cell line.
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同义词——
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通路Cytoskeleton/Cell Adhesion Molecules
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靶点Kinesin
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受体Kinesin
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研究领域——
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适应症——
化学信息
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CAS Number912953-25-4
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分子量291.27
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分子式C16H12F3NO
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纯度>98% (HPLC)
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溶解度——
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SMILESC1CC(=O)NC2=C1C=C(C=C2)C3=CC=C(C=C3)C(F)(F)F
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化学全称6-(4-(trifluoromethyl)phenyl)-3,4-dihydroquinolin-2(1H)-one
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1. Luo L, et al. Nat Chem Biol. 2007 Nov;3(11):722-6.
产品手册
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GSK-1
GSK-1 is an ATP-competitive inhibitor of the mitotic kinesin KSP with HCT116 cell IC50 of 36 nM.