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CGK-1026
CAS No. 287383-59-9
CGK-1026 ( CGK 1026;CGK1026 )
产品货号. M13877 CAS No. 287383-59-9
A small molecule that inhibits human telomerase reverse transcriptase (hTERT) expression.
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| 规格 | 价格/人民币 | 库存 | 数量 |
| 5MG | ￥527 | 有现货 |
|
| 10MG | ￥794 | 有现货 |
|
| 25MG | ￥1742 | 有现货 |
|
| 50MG | ￥3216 | 有现货 |
|
| 100MG | ￥4836 | 有现货 |
|
| 500MG | ￥10206 | 有现货 |
|
| 1G | 获取报价 | 有现货 |
|
生物学信息
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产品名称CGK-1026
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注意事项本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
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产品简述A small molecule that inhibits human telomerase reverse transcriptase (hTERT) expression.
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产品描述A small molecule that inhibits human telomerase reverse transcriptase (hTERT) expression; inhibits the recruitment of HDAC into E2F-pocket protein complexes assembled on the hTERT promoter, inhibits HDAC activity with IC50 of 100 nM; induces G1 arrest of IMR90 cells.
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同义词CGK 1026;CGK1026
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通路Cell Cycle/DNA Damage
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靶点HDAC
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受体HDAC
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研究领域Cancer
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适应症——
化学信息
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CAS Number287383-59-9
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分子量326.35
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分子式C18H18N2O4
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纯度>98% (HPLC)
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溶解度DMSO: 32.6 mg/mL (100 mM) （ < 1 mg/ml refers to the product slightly soluble or insoluble )
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SMILESO=C(NO)CCCCCN(C(C1=CC=CC2=CC=CC3=C12)=O)C3=O
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化学全称N-Hydroxy-1,3-dioxo-1H-benz[de]isoquinoline-2(3H)-hexanamide
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1. Won J, et al. Proc Natl Acad Sci U S A. 2004 Aug 3;101(31):11328-33.
2. Alimirah F, et al. Mol Cancer Res. 2007 Mar;5(3):251-9.
3. Song LL, et al. PLoS One. 2010 Jan 5;5(1):e8569.
2. Alimirah F, et al. Mol Cancer Res. 2007 Mar;5(3):251-9.
3. Song LL, et al. PLoS One. 2010 Jan 5;5(1):e8569.
产品手册
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