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Temanogrel
CAS No. 887936-68-7
Temanogrel ( APD791 )
产品货号. M24910 CAS No. 887936-68-7
Temanogrel is a highly selective antagonist of the 5-HT2A receptor (Ki: 4.9 nM).
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| 规格 | 价格/人民币 | 库存 | 数量 |
| 5MG | ￥2130 | 有现货 |
|
| 10MG | ￥3183 | 有现货 |
|
| 25MG | ￥5330 | 有现货 |
|
| 50MG | ￥7590 | 有现货 |
|
| 100MG | ￥10287 | 有现货 |
|
| 200MG | 获取报价 | 有现货 |
|
| 500MG | 获取报价 | 有现货 |
|
| 1G | 获取报价 | 有现货 |
|
生物学信息
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产品名称Temanogrel
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注意事项本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
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产品简述Temanogrel is a highly selective antagonist of the 5-HT2A receptor (Ki: 4.9 nM).
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产品描述Temanogrel is a highly selective antagonist of the 5-HT2A receptor (Ki: 4.9 nM).
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同义词APD791
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通路Endocrinology/Hormones
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靶点5-HT Receptor
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受体5-HT2A
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研究领域——
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适应症——
化学信息
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CAS Number887936-68-7
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分子量436.5
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分子式C24H28N4O4
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纯度>98% (HPLC)
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溶解度DMSO:125 mg/mL (286.37 mM; Need ultrasonic)
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SMILESCn1nccc1-c(cc(cc1)NC(c2cc(OC)ccc2)=O)c1OCCN1CCOCC1
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化学全称——
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1.Xiong Y, et al. Discovery and structure-activity relationship of 3-methoxy-N-(3-(1-methyl-1H-pyrazol-5-yl)-4-(2-morpholinoethoxy)phenyl)benzamide (APD791): a highly selective 5-hydroxytryptamine2A receptor inverse agonist for the treatment of arterial thrombosis. J Med Chem. 2010 Jun 10;53(11):4412-21.
产品手册
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