Temanogrel
CAS No. 887936-68-7
Temanogrel ( APD791 )
产品货号. M24910 CAS No. 887936-68-7
Temanogrel is a highly selective antagonist of the 5-HT2A receptor (Ki: 4.9 nM).
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
规格 | 价格/人民币 | 库存 | 数量 |
5MG | ¥2130 | 有现货 |
|
10MG | ¥3183 | 有现货 |
|
25MG | ¥5330 | 有现货 |
|
50MG | ¥7590 | 有现货 |
|
100MG | ¥10287 | 有现货 |
|
200MG | 获取报价 | 有现货 |
|
500MG | 获取报价 | 有现货 |
|
1G | 获取报价 | 有现货 |
|
生物学信息
-
产品名称Temanogrel
-
注意事项本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
-
产品简述Temanogrel is a highly selective antagonist of the 5-HT2A receptor (Ki: 4.9 nM).
-
产品描述Temanogrel is a highly selective antagonist of the 5-HT2A receptor (Ki: 4.9 nM).
-
同义词APD791
-
通路Endocrinology/Hormones
-
靶点5-HT Receptor
-
受体5-HT2A
-
研究领域——
-
适应症——
化学信息
-
CAS Number887936-68-7
-
分子量436.5
-
分子式C24H28N4O4
-
纯度>98% (HPLC)
-
溶解度DMSO:125 mg/mL (286.37 mM; Need ultrasonic)
-
SMILESCn1nccc1-c(cc(cc1)NC(c2cc(OC)ccc2)=O)c1OCCN1CCOCC1
-
化学全称——
运输与储存
-
储存条件(-20℃)
-
运输条件With Ice Pack
-
稳定性≥ 2 years
参考文献
1.Xiong Y, et al. Discovery and structure-activity relationship of 3-methoxy-N-(3-(1-methyl-1H-pyrazol-5-yl)-4-(2-morpholinoethoxy)phenyl)benzamide (APD791): a highly selective 5-hydroxytryptamine2A receptor inverse agonist for the treatment of arterial thrombosis. J Med Chem. 2010 Jun 10;53(11):4412-21.
产品手册
关联产品
-
Doxepin hydrochlorid...
Doxepin HCl is a tricyclic antidepressant that is marketed worldwide.
-
Nefazodone hydrochlo...
Nefazodone hydrochloride is an antidepressant drug.
-
N-Acetyl-5-hydroxytr...
N-Acetylserotonin (NAS), also known as normelatonin, is a naturally occurring chemical intermediate in the endogenous production of melatonin from serotonin.