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Ritanserin
CAS No. 87051-43-2
Ritanserin ( R 55667 )
产品货号. M24881 CAS No. 87051-43-2
Ritanserin is a highly effective, relatively selective, long-acting antagonist of 5-HT2 receptor (IC50: 0.9 nM), less active on Histamine H1, Dopamine D2, Adrenergic α1, Adrenergic α2 receptors.
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| 规格 | 价格/人民币 | 库存 | 数量 |
| 2MG | ￥389 | 有现货 |
|
| 5MG | ￥624 | 有现货 |
|
| 10MG | ￥940 | 有现货 |
|
| 25MG | ￥1580 | 有现货 |
|
| 50MG | ￥2333 | 有现货 |
|
| 100MG | ￥3507 | 有现货 |
|
| 200MG | 获取报价 | 有现货 |
|
| 500MG | 获取报价 | 有现货 |
|
| 1G | 获取报价 | 有现货 |
|
生物学信息
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产品名称Ritanserin
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注意事项本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
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产品简述Ritanserin is a highly effective, relatively selective, long-acting antagonist of 5-HT2 receptor (IC50: 0.9 nM), less active on Histamine H1, Dopamine D2, Adrenergic α1, Adrenergic α2 receptors.
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产品描述Ritanserin is a highly effective, relatively selective, long-acting antagonist of 5-HT2 receptor (IC50: 0.9 nM), less active on Histamine H1, Dopamine D2, Adrenergic α1, Adrenergic α2 receptors.
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同义词R 55667
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通路Endocrinology/Hormones
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靶点5-HT Receptor
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受体5-HT2;D2;H1 receptor;α1-adrenergic receptor;α2 receptor
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研究领域——
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适应症——
化学信息
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CAS Number87051-43-2
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分子量477.6
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分子式C27H25F2N3OS
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纯度>98% (HPLC)
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溶解度DMSO:25 mg/mL (52.35 mM; Need ultrasonic)
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SMILESCC1=C(C(N(C=CS2)C2=N1)=O)CCN(CC/3)CCC3=C(C4=CC=C(F)C=C4)\C5=CC=C(F)C=C5
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化学全称——
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1.Leysen JE, et al. Receptor-binding properties in vitro and in vivo of ritanserin: A very potent and long acting serotonin-S2 antagonist. Mol Pharmacol. 1985 Jun;27(6):600-11.
产品手册
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