Ralaniten
CAS No. 1203490-23-6
Ralaniten ( EPI-506 )
产品货号. M10744 CAS No. 1203490-23-6
Ralaniten (EPI-506) is a novel small-molecule inhibitor of androgen receptor (AR) N-terminal domain inhibitor for the treatment of advanced prostate cancer.
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
规格 | 价格/人民币 | 库存 | 数量 |
50MG | ¥3345 | 有现货 |
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100MG | ¥5370 | 有现货 |
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200MG | 获取报价 | 有现货 |
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500MG | 获取报价 | 有现货 |
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1G | 获取报价 | 有现货 |
|
生物学信息
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产品名称Ralaniten
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注意事项本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
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产品简述Ralaniten (EPI-506) is a novel small-molecule inhibitor of androgen receptor (AR) N-terminal domain inhibitor for the treatment of advanced prostate cancer.
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产品描述Ralaniten (EPI-506) is a novel small-molecule inhibitor of androgen receptor (AR) N-terminal domain inhibitor for the treatment of advanced prostate cancer; AR NTD-targeting agents have the potential to overcome shortcomings of current hormonal therapies by inhibiting all forms of AR-mediated transcriptional activity, and as a result, may affect a broader AR population including mutational and splice variant ARs.Prostate Cancer Phase 2 Clinical
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同义词EPI-506
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通路Endocrinology/Hormones
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靶点Estrogen Receptor/ERR
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受体Estrogen Receptor/ERR
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研究领域Cancer
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适应症Prostate Cancer
化学信息
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CAS Number1203490-23-6
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分子量394.89
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分子式C21H27ClO5
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纯度>98% (HPLC)
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溶解度——
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SMILESCC(C)(C1=CC=C(C=C1)OCC(CO)O)C2=CC=C(C=C2)OCC(CCl)O
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化学全称(2R)-3-[4-(2-{4-[(2S)-3-chloro- 2-hydroxypropoxy]phenyl}propan-2-yl)phenoxy]propane- 1,2-diol
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1. Antonarakis ES, et al. Oncologist. 2016 Dec;21(12):1427-1435.
产品手册
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