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R-7128

CAS No. 940908-79-2

R-7128 ( RG-7128;Mericitabine;PSI-6130 diisobutyrate )

产品货号. M16730 CAS No. 940908-79-2

The prodrug of PSI-6130, a potent, specific inhibitor of HCV RNA synthesis by inhibiting the NS5B RNA polymerase.

纯度: >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
规格 价格/人民币 库存 数量
5MG ¥1482 有现货
10MG ¥2066 有现货
25MG ¥3572 有现货
50MG ¥5257 有现货
100MG ¥7501 有现货
500MG ¥15147 有现货
1G 获取报价 有现货

生物学信息

  • 产品名称
    R-7128
  • 注意事项
    本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
  • 产品简述
    The prodrug of PSI-6130, a potent, specific inhibitor of HCV RNA synthesis by inhibiting the NS5B RNA polymerase.
  • 产品描述
    The prodrug of PSI-6130, a potent, specific inhibitor of HCV RNA synthesis by inhibiting the NS5B RNA polymerase.HCV Infection Phase 2 Discontinued
  • 同义词
    RG-7128;Mericitabine;PSI-6130 diisobutyrate
  • 通路
    Microbiology/Virology
  • 靶点
    HCV
  • 受体
    HCV
  • 研究领域
    Infection
  • 适应症
    HCV Infection

化学信息

  • CAS Number
    940908-79-2
  • 分子量
    399.41
  • 分子式
    C18H26FN3O6
  • 纯度
    >98% (HPLC)
  • 溶解度
    10 mM in DMSO
  • SMILES
    O=C(N=C(C=C1)N)N1[C@H](O2)[C@](C)(F)[C@H](OC(C(C)C)=O)[C@H]2COC(C(C)C)=O
  • 化学全称
    Cytidine, 2'-deoxy-2'-fluoro-2'-methyl-, 3',5'-bis(2-methylpropanoate), (2'R)-

运输与储存

  • 储存条件
    (-20℃)
  • 运输条件
    With Ice Pack
  • 稳定性
    ≥ 2 years

参考文献

1. McCown MF, et al. Antimicrob Agents Chemother. 2008 May;52(5):1604-12.
2. Ali S, et al. Antimicrob Agents Chemother. 2008 Dec;52(12):4356-69.
3. Le Pogam S, et al. J Infect Dis. 2010 Nov 15;202(10):1510-9.
4. Guedj J, et al. Hepatology. 2012 Apr;55(4):1030-7.
产品手册
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