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首页- Products - Endocrinology/Hormones - 5-HT Receptor - Pimethixene

Pimethixene

CAS No. 314-03-4

Pimethixene ( Pimetixene; Calmixen )

产品货号. M24244 CAS No. 314-03-4

Pimethixene is a highly potent 5-HT1A, 5-HT2A, 5-HT2B, 5-HT2C, histamine H1, dopamine D2 and D4.4 as well as muscarinic M1 and M2 receptors antagonist(pKis of 7.63, 10.22, 10.44, 8.42, 10.14, 8.19, 7.54, 8.61 and 9.38, respectively).

纯度: >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
规格 价格/人民币 库存 数量
2MG ￥389 有现货
5MG ￥575 有现货
10MG ￥818 有现货
25MG ￥1458 有现货
50MG ￥2163 有现货
100MG ￥3216 有现货
200MG ￥4803 有现货
500MG ￥7687 有现货
1G 获取报价 有现货
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生物学信息

  • 产品名称
    Pimethixene
  • 注意事项
    本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
  • 产品简述
    Pimethixene is a highly potent 5-HT1A, 5-HT2A, 5-HT2B, 5-HT2C, histamine H1, dopamine D2 and D4.4 as well as muscarinic M1 and M2 receptors antagonist(pKis of 7.63, 10.22, 10.44, 8.42, 10.14, 8.19, 7.54, 8.61 and 9.38, respectively).
  • 产品描述
    Pimethixene is a highly potent 5-HT1A, 5-HT2A, 5-HT2B, 5-HT2C, histamine H1, dopamine D2 and D4.4 as well as muscarinic M1 and M2 receptors antagonist(pKis of 7.63, 10.22, 10.44, 8.42, 10.14, 8.19, 7.54, 8.61 and 9.38, respectively).
  • 同义词
    Pimetixene; Calmixen
  • 通路
    Endocrinology/Hormones
  • 靶点
    5-HT Receptor
  • 受体
    5-HT2A Receptor;5-HT2B Receptor;5-HT2C Receptor;H1 receptor;5-HT1A Receptor;D2 receptor;DD4.4 receptor;M1 receptor;M2 receptor
  • 研究领域
    ——
  • 适应症
    ——

化学信息

  • CAS Number
    314-03-4
  • 分子量
    293.4
  • 分子式
    C19H19NS
  • 纯度
    >98% (HPLC)
  • 溶解度
    ——
  • SMILES
    CN(CC1)CCC1=C1c(cccc2)c2Sc2c1cccc2
  • 化学全称
    ——

运输与储存

  • 储存条件
    (-20℃)
  • 运输条件
    With Ice Pack
  • 稳定性
    ≥ 2 years

参考文献

1.Schmitz B, et al. BF-1--a novel selective 5-HT2B receptor antagonist blocking neurogenic dural plasma protein extravasation in guinea pigs. Eur J Pharmacol. 2015 Mar 15;751:73-80.
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