PRX-08066
CAS No. 866206-54-4
PRX-08066 ( —— )
产品货号. M24869 CAS No. 866206-54-4
PRX-08066 is a selective 5-hydroxytryptamine receptor 2B (5-HT2BR, IC50= 3.4 nM) antagonist that induces selective vasodilation of pulmonary arteries.
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
规格 | 价格/人民币 | 库存 | 数量 |
5MG | ¥988 | 有现货 |
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10MG | ¥1442 | 有现货 |
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25MG | ¥2989 | 有现货 |
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50MG | ¥4447 | 有现货 |
|
100MG | ¥6383 | 有现货 |
|
500MG | ¥13203 | 有现货 |
|
1G | 获取报价 | 有现货 |
|
生物学信息
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产品名称PRX-08066
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注意事项本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
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产品简述PRX-08066 is a selective 5-hydroxytryptamine receptor 2B (5-HT2BR, IC50= 3.4 nM) antagonist that induces selective vasodilation of pulmonary arteries.
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产品描述PRX-08066 is a selective 5-hydroxytryptamine receptor 2B (5-HT2BR, IC50= 3.4 nM) antagonist that induces selective vasodilation of pulmonary arteries.
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同义词——
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通路Endocrinology/Hormones
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靶点5-HT Receptor
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受体5-HT2B
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研究领域——
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适应症——
化学信息
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CAS Number866206-54-4
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分子量401.9
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分子式C19H17ClFN5S
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纯度>98% (HPLC)
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溶解度DMSO:7 mg/mL (17.42 mM; Need ultrasonic)
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SMILESC1CN(CCC1NC2=C3C=C(SC3=NC=N2)Cl)CC4=CC(=C(C=C4)F)C#N
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化学全称——
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1.Porvasnik SL, et al. PRX-08066, a novel 5-hydroxytryptamine receptor 2B antagonist, reduces monocrotaline-induced pulmonary arterial hypertension and right ventricular hypertrophy in rats. J Pharmacol Exp Ther. 2010 Aug;334(2):364-72.
产品手册
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