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PFI-4
CAS No. 900305-37-5
PFI-4 ( PFI-4; PFI 4; PFI4 )
产品货号. M16470 CAS No. 900305-37-5
A potent, selective inhibitor of the BRPF1 bromodomain with pIC50 of 7.3.
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| 规格 | 价格/人民币 | 库存 | 数量 |
| 5MG | ￥486 | 有现货 |
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| 10MG | ￥640 | 有现货 |
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| 25MG | ￥1312 | 有现货 |
|
| 50MG | ￥2552 | 有现货 |
|
| 100MG | ￥4455 | 有现货 |
|
| 200MG | 获取报价 | 有现货 |
|
| 500MG | 获取报价 | 有现货 |
|
| 1G | 获取报价 | 有现货 |
|
生物学信息
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产品名称PFI-4
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注意事项本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
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产品简述A potent, selective inhibitor of the BRPF1 bromodomain with pIC50 of 7.3.
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产品描述A potent, selective inhibitor of the BRPF1 bromodomain with pIC50 of 7.3; exhibits >100-fold selectivity for BRPF1 over a panel of other bromodomains including BRPF2 (BRD1), BRPF3 and BRD4.
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同义词PFI-4; PFI 4; PFI4
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通路Chromatin/Epigenetic
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靶点Bromodomain
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受体BRPF1;BRPF2;BRPF3
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研究领域Other Indications
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适应症——
化学信息
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CAS Number900305-37-5
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分子量380.44
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分子式C21H24N4O3
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纯度>98% (HPLC)
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溶解度DMSO: 26 mg/mL
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SMILESO=C(NC1=C(N2CCCC2)C=C(N3C)C(N(C)C3=O)=C1)C4=CC=CC=C4OC
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化学全称Benzamide, N-[2,3-dihydro-1,3-dimethyl-2-oxo-6-(1-pyrrolidinyl)-1H-benzimidazol-5-yl]-2-methoxy-
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1. Demont EH, et al. ACS Med Chem Lett. 2014 Sep 10;5(11):1190-5.
产品手册
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