BRPF1-IN-3
CAS No. 901245-65-6
BRPF1-IN-3 ( GSK-5959; GSK 5959; GSK5959. )
产品货号. M16481 CAS No. 901245-65-6
BRPF1-IN-3 is a potent, selective, membrane permeable BRPF1 bromodomain inhibitor with pIC50 of 7.1.
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
规格 | 价格/人民币 | 库存 | 数量 |
5MG | ¥421 | 有现货 |
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10MG | ¥721 | 有现货 |
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25MG | ¥1288 | 有现货 |
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50MG | ¥2130 | 有现货 |
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100MG | ¥3175 | 有现货 |
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200MG | ¥4641 | 有现货 |
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500MG | 获取报价 | 有现货 |
|
1G | 获取报价 | 有现货 |
|
生物学信息
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产品名称BRPF1-IN-3
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注意事项本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
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产品简述BRPF1-IN-3 is a potent, selective, membrane permeable BRPF1 bromodomain inhibitor with pIC50 of 7.1.
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产品描述BRPF1-IN-3 is a potent, selective, membrane permeable BRPF1 bromodomain inhibitor with pIC50 of 7.1; shows 100- and >1000-fold selectivity over BRPF2 and BRPF3, respectively; exhibits an IC50 of 0.98 uM in cellular protein interaction assay (displacement of NanoLuc-tagged BRPF1 bromodomain from Halo-tagged histone H3.3).
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同义词GSK-5959; GSK 5959; GSK5959.
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通路Chromatin/Epigenetic
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靶点Bromodomain
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受体BRPF1
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研究领域Other Indications
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适应症——
化学信息
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CAS Number901245-65-6
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分子量394.48
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分子式C22H26N4O3
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纯度>98% (HPLC)
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溶解度DMSO: 10 mM ( < 1 mg/ml refers to the product slightly soluble or insoluble )
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SMILESO=C(NC1=C(N2CCCCC2)C=C(N3C)C(N(C)C3=O)=C1)C4=CC=CC=C4OC
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化学全称N-(1,3-dimethyl-2-oxo-6-(piperidin-1-yl)-2,3-dihydro-1H-benzo[d]imidazol-5-yl)-2-methoxybenzamide
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
产品手册
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