PF-04995274 ( PF-4995274;TBPT )

产品货号. M11321 CAS No. 1331782-27-4

COA

Datasheet

HNMR

HPLC

MSDS

Handing Instructions

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产品名称

PF-04995274
注意事项

本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
产品简述

PF-04995274 (TBPT) is a novel potent, sellective, partial agonist of 5-HT4 receptor under investigation for neurological disorders.
产品描述

PF-04995274 (TBPT) is a novel potent, sellective, partial agonist of 5-HT4 receptor under investigation for neurological disorders.Alzheimer Disease Phase 1 Discontinued
同义词

PF-4995274;TBPT
通路

Endocrinology/Hormones
靶点

5-HT Receptor
受体

5-HT Receptor
研究领域

Neurological Disease
适应症

Alzheimer Disease

CAS Number

1331782-27-4
分子量

432.52
分子式

C23H32N2O6
纯度

>98% (HPLC)
溶解度

——
SMILES

C1CN(CCC1COC2=NOC3=C2C(=CC=C3)OC4CCOC4)CC5(CCOCC5)O
化学全称

(R)-4-((4-(((4-(Tetrahydrofuran-3-yloxy)-1,2-benzisoxazol-3-yl)oxy)methyl)piperidin-1-yl)methyl)tetrahydro-2H-pyran-4-ol

1. Sawant-Basak A, et al. J Pharm Sci. 2013 Sep;102(9):3277-93.

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