Mestranol ( EE 3-ME; Ethynyl Estradiol 3-methyl ether; NSC 84032; SC-475; Δ-MVE )

产品货号. M15769 CAS No. 72-33-3

COA

Datasheet

HNMR

HPLC

MSDS

Handing Instructions

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产品名称

Mestranol
注意事项

本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
产品简述

Mestranol is the 3-methyl ether of ethinylestradiol. It was the estrogen used in many of the first oral contraceptives.
产品描述

Mestranol is the 3-methyl ether of ethinylestradiol. It was the estrogen used in many of the first oral contraceptives. It is a biologically inactive prodrug of ethinylestradiol to which it is demethylated in the liver with a conversion efficiency of 70%.
同义词

EE 3-ME; Ethynyl Estradiol 3-methyl ether; NSC 84032; SC-475; Δ-MVE
通路

Endocrinology/Hormones
靶点

Estrogen Receptor/ERR
受体

ER
研究领域

Endocrinology
适应症

——

CAS Number

72-33-3
分子量

310.43
分子式

C21H26O2
纯度

>98%(HPLC)
溶解度

Ethanol: 25 mg/mL (80.53 mM); DMSO: 15 mg/mL (48.32 mM)
SMILES

CC12CCC3C(C1CCC2(C#C)O)CCC4=C3C=CC(=C4)OC
化学全称

17-ethynyl-3-methoxy-13-methyl-7,8,9,11,12,13,14,15,16,17-decahydro-6H-cyclopenta[a]phenanthren-17-ol

1.IARC Monogr Eval Carcinog Risk Chem Hum. 1979 Dec;21:257-78.

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