• 咨询热线
    客服服务热线 13671568941/15317326293
  • 在线咨询
  • 微信客服
    微信客服
  • 公众号
    扫码关注公众号

GSK5182

CAS No. 877387-37-6

GSK5182 ( —— )

产品货号. M21654 CAS No. 877387-37-6

GSK5182 is a highly selective inverse estrogen-related receptor γ agonist (IC50 : 79 nM)?.

纯度: >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
规格 价格/人民币 库存 数量
2MG ¥551 有现货
5MG ¥786 有现货
10MG ¥1256 有现货
25MG ¥2341 有现货
50MG ¥3548 有现货
100MG ¥5241 有现货
200MG 获取报价 有现货
500MG 获取报价 有现货
1G 获取报价 有现货

生物学信息

  • 产品名称
    GSK5182
  • 注意事项
    本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
  • 产品简述
    GSK5182 is a highly selective inverse estrogen-related receptor γ agonist (IC50 : 79 nM)?.
  • 产品描述
    GSK5182 is a highly selective inverse estrogen-related receptor γ agonist (IC50 : 79 nM)?.
  • 同义词
    ——
  • 通路
    Endocrinology/Hormones
  • 靶点
    Estrogen Receptor/ERR
  • 受体
    ERRγ
  • 研究领域
    ——
  • 适应症
    ——

化学信息

  • CAS Number
    877387-37-6
  • 分子量
    417.55
  • 分子式
    C27H31NO3
  • 纯度
    >98% (HPLC)
  • 溶解度
    ——
  • SMILES
    CN(C)CCOc1ccc(cc1)C(\c1ccc(O)cc1)=C(\CCCO)c1ccccc1
  • 化学全称
    4-[(Z)-1-[4-(2-dimethylaminoethoxy)phenyl]-5-hydroxy-2-phenylpent-1-enyl]phenol

运输与储存

  • 储存条件
    (-20℃)
  • 运输条件
    With Ice Pack
  • 稳定性
    ≥ 2 years

参考文献

1.Kim JH et al. Estrogen-related receptor γ is upregulated in liver cancer and its inhibition suppresses livercancer cell proliferation via induction of p21 and p27. Exp Mol Med. 2016 Mar 4;48:e213.
产品手册
关联产品
  • Diarylpropionitrile

    Diarylpropionitrile (DPN) is a non-steroidal estrogen receptor β(ERβ) selective ligand.

  • Endoxifen hydrochlor...

    A metabolite of tamoxifen, orally active non-steroidal selective estrogen receptor modulator (SERM) for the treatment of estrogen receptor-positive breast cancer.

  • Enclomiphene citrate

    Enclomiphene citrate((E)-Clomifene, cis-Clomifene, RMI-16289, ICI-46476)is a nonsteroidal selective estrogen receptor modulator (SERM) that is under development for the treatment of male hypogonadism.