GSK854 ( —— )

产品货号. M33986 CAS No. 1316059-00-3

COA

Datasheet

HNMR

HPLC

MSDS

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产品名称

GSK854
注意事项

本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
产品简述

GSK854 是一种有效的肌钙蛋白 I 相互作用激酶 (TNNI3K) 抑制剂。GSK854 是一种合适的先导活性分子，可用于识别新的心脏活性分子，并已在旨在确定 TNNI3K 在心力衰竭中的作用的研究中用作体内工具。
产品描述

GSK854 is a potent Inhibitor of Troponin I-Interacting Kinase (TNNI3K). GSK854 is a suitable lead for identifying new cardiac medicines and have been employed as in vivo tools in investigational studies aimed at defining the role of TNNI3K within heart failure.
体外实验

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体内实验

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同义词

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通路

Apoptosis
靶点

Apoptosis
受体

Apoptosis
研究领域

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适应症

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1. Philp J, et al. 4,6-Diaminopyrimidines as Highly Preferred Troponin I-Interacting Kinase (TNNI3K) Inhibitors. J Med Chem. 2018;61(7):3076-3088.?

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