Bilastine ( Bilastine trade name Bilaxten )

产品货号. M18206 CAS No. 202189-78-4

比拉斯汀是一种新型新一代抗组胺药，对H1组胺受体具有高度选择性，起效快，作用持续时间长。

纯度: >98% (HPLC)

COA

Datasheet

HNMR

HPLC

MSDS

Handing Instructions

规格	价格/人民币	库存	数量
2MG	￥119	有现货
5MG	￥177	有现货
10MG	￥245	有现货
25MG	￥384	有现货
50MG	￥616	有现货
100MG	￥963	有现货
500MG	￥2187	有现货
1G	获取报价	有现货
1 mL x 10 mM in DMSO	￥240	有现货

产品询价大包装询价加入购物车

生物学信息

产品名称

Bilastine
注意事项

本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
产品简述

比拉斯汀是一种新型新一代抗组胺药，对H1组胺受体具有高度选择性，起效快，作用持续时间长。
产品描述

Bilastine (trade name Bilaxten) is a second generation antihistamine drug for the treatment of allergic rhinoconjunctivitis and urticaria (hives). It exerts its effect as a selective histamine H1 receptor antagonist, and has a potency similar to cetirizine and is superior to fexofenadine. It was developed in Spain by FAES Farma. Bilastine is approved in the European Union for the symptomatic treatment of allergic rhinoconjunctivitis and urticaria, but it is not approved by the U.S. Food and Drug Administration for any use in the United States. Bilastine has been effective in the treatment of ocular symptoms and diseases of allergies, including rhinoconjuctivitis. Additionally, bilastine has been shown to improve quality of life, and all nasal and ocular symptoms related to allergic rhinitis.
体外实验

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体内实验

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同义词

Bilastine trade name Bilaxten
通路

Endocrinology/Hormones
靶点

5-HT Receptor
受体

H1 receptor
研究领域

Inflammation/Immunology
适应症

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化学信息

CAS Number

202189-78-4
分子量

463.62
分子式

C28H37N3O3
纯度

>98% (HPLC)
溶解度

DMSO : ≥ 49.3 mg/mL; 106.34 mM
SMILES

CCOCCn1c(nc2ccccc12)C1CCN(CCc2ccc(cc2)C(C)(C)C(O)=O)CC1
化学全称

2-(4-(2-(4-(1-(2-ethoxyethyl)-1H-benzo[d]imidazol-2-yl)piperidin-1-yl)ethyl)phenyl)-2-methylpropanoic acid

运输与储存

储存条件

(-20℃)
运输条件

With Ice Pack
稳定性

≥ 2 years

参考文献

1.Wolthers OD.Bilastine: a new nonsedating oral H1 antihistamine for treatment of allergic rhinoconjunctivitis and urticaria.Biomed Res Int. 2013;2013:626837.

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