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Gestrinone
CAS No. 16320-04-0
Gestrinone ( R 2323 )
产品货号. M20652 CAS No. 16320-04-0
Gestrinone is a synthetic androgen receptor agonist and ER and progesterone receptor antagonist used to treat endometriosis.
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| 规格 | 价格/人民币 | 库存 | 数量 |
| 5MG | ￥503 | 有现货 |
|
| 10MG | ￥811 | 有现货 |
|
| 25MG | ￥1455 | 有现货 |
|
| 50MG | ￥2187 | 有现货 |
|
| 100MG | 获取报价 | 有现货 |
|
| 200MG | 获取报价 | 有现货 |
|
| 500MG | 获取报价 | 有现货 |
|
| 1G | 获取报价 | 有现货 |
|
生物学信息
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产品名称Gestrinone
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注意事项本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
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产品简述Gestrinone is a synthetic androgen receptor agonist and ER and progesterone receptor antagonist used to treat endometriosis.
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产品描述Gestrinone is a synthetic androgen receptor agonist and ER and progesterone receptor antagonist used to treat endometriosis. It inhibits leiomyoma cells with an IC50 of 43.67 μM.
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同义词R 2323
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通路Endocrinology/Hormones
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靶点Estrogen Receptor/ERR
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受体ER
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研究领域Others
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适应症Endometriosis with or without accompanying sterility
化学信息
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CAS Number16320-04-0
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分子量308.41
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分子式C21H24O2
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纯度>98% (HPLC)
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溶解度DMSO:50 mg/mL (162.12 mM)
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SMILES[H][C@@]12CC[C@@](O)(C#C)[C@@]1(CC)C=CC1=C3CCC(=O)C=C3CC[C@@]21[H]
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化学全称(8S13S14S17S)-13-ethyl-17-ethynyl-17-hydroxy-126781314151617-decahydro-3H-cyclopenta[a]phenanthren-3-one
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1.Hui-Ling X Ning Y Jing W et al. Therapeutic effects of mifepristone combined withGestrinone on patients with endometriosis[J]. Pakistan Journal of Medical Sciences 2016 32(5).
产品手册
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