021-51111890
购物车（）
sales@molnova.cn
Gestrinone
CAS No. 16320-04-0
Gestrinone ( R 2323 )
产品货号. M20652 CAS No. 16320-04-0
Gestrinone is a synthetic androgen receptor agonist and ER and progesterone receptor antagonist used to treat endometriosis.
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| 规格 | 价格/人民币 | 库存 | 数量 |
| 5MG | ￥503 | 有现货 |
|
| 10MG | ￥811 | 有现货 |
|
| 25MG | ￥1455 | 有现货 |
|
| 50MG | ￥2187 | 有现货 |
|
| 100MG | 获取报价 | 有现货 |
|
| 200MG | 获取报价 | 有现货 |
|
| 500MG | 获取报价 | 有现货 |
|
| 1G | 获取报价 | 有现货 |
|
生物学信息
-
产品名称Gestrinone
-
注意事项本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
-
产品简述Gestrinone is a synthetic androgen receptor agonist and ER and progesterone receptor antagonist used to treat endometriosis.
-
产品描述Gestrinone is a synthetic androgen receptor agonist and ER and progesterone receptor antagonist used to treat endometriosis. It inhibits leiomyoma cells with an IC50 of 43.67 μM.
-
同义词R 2323
-
通路Endocrinology/Hormones
-
靶点Estrogen Receptor/ERR
-
受体ER
-
研究领域Others
-
适应症Endometriosis with or without accompanying sterility
化学信息
-
CAS Number16320-04-0
-
分子量308.41
-
分子式C21H24O2
-
纯度>98% (HPLC)
-
溶解度DMSO:50 mg/mL (162.12 mM)
-
SMILES[H][C@@]12CC[C@@](O)(C#C)[C@@]1(CC)C=CC1=C3CCC(=O)C=C3CC[C@@]21[H]
-
化学全称(8S13S14S17S)-13-ethyl-17-ethynyl-17-hydroxy-126781314151617-decahydro-3H-cyclopenta[a]phenanthren-3-one
运输与储存
-
储存条件(-20℃)
-
运输条件With Ice Pack
-
稳定性≥ 2 years
参考文献
1.Hui-Ling X Ning Y Jing W et al. Therapeutic effects of mifepristone combined withGestrinone on patients with endometriosis[J]. Pakistan Journal of Medical Sciences 2016 32(5).
产品手册
关联产品
-
Chrysin
Chrysin is mainly found in passion flowers, honey, and propolis acts as a potential therapeutic and preventive agent to inhibit proliferation and invasion of various human cancer cells.
-
Acolbifene
Acolbifene is a selective antagonist of estrogen receptors with IC50s of 2 nM and 0.4 nM for estradiol-induced transcriptional activity of ERα and ERβ. Acolbifene shows an anticarcinogenic property.
-
Diarylpropionitrile
Diarylpropionitrile (DPN) is a non-steroidal estrogen receptor β(ERβ) selective ligand.
