GSK525768A
CAS No. 1260530-25-3
GSK525768A ( GSK 525768A;GSK-525768A )
产品货号. M11076 CAS No. 1260530-25-3
GSK525768A is an enantiomer, negative control compound of I-BET762 (GSK525762A).
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
规格 | 价格/人民币 | 库存 | 数量 |
5MG | ¥2811 | 有现货 |
|
50MG | ¥12393 | 有现货 |
|
100MG | ¥16119 | 有现货 |
|
200MG | 获取报价 | 有现货 |
|
500MG | 获取报价 | 有现货 |
|
1G | 获取报价 | 有现货 |
|
生物学信息
-
产品名称GSK525768A
-
注意事项本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
-
产品简述GSK525768A is an enantiomer, negative control compound of I-BET762 (GSK525762A).
-
产品描述GSK525768A is an enantiomer, negative control compound of I-BET762 (GSK525762A), shows no activity against BET family proteins BRD2, BRD3 and BRD4.
-
同义词GSK 525768A;GSK-525768A
-
通路Chromatin/Epigenetic
-
靶点Bromodomain
-
受体Bromodomain
-
研究领域Inflammation/Immunology
-
适应症——
化学信息
-
CAS Number1260530-25-3
-
分子量423.90
-
分子式C22H22ClN5O2
-
纯度>98% (HPLC)
-
溶解度10 mM in DMSO
-
SMILESCCNC(=O)CC1C2=NN=C(N2C3=C(C=C(C=C3)OC)C(=N1)C4=CC=C(C=C4)Cl)C
-
化学全称4H-[1,2,4]Triazolo[4,3-a][1,4]benzodiazepine-4-acetamide, 6-(4-chlorophenyl)-N-ethyl-8-methoxy-1-methyl-, (4R)-
运输与储存
-
储存条件(-20℃)
-
运输条件With Ice Pack
-
稳定性≥ 2 years
参考文献
1. Nicodeme E, et al. Nature. 2010 Dec 23;468(7327):1119-23.
产品手册
关联产品
-
TP-238
TP-238 (TP238) is a CECR2/BPTF bromodomains chemical probe with IC50 of 30nM against CECR2 and 350nM against BPTF in an alphascreen assay.
-
GW 841819X
GW 841819X is an analogue of (+)-JQ1 and a novel inhibitor of BET bromodomain.
-
CPI-637
A potent and selective, cell-active CBP/EP300 bromodomain inhibitor with CBP BRET EC50 of 0.03 uM.