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首页- Products - Chromatin/Epigenetic - Bromodomain - GSK525768A

GSK525768A

CAS No. 1260530-25-3

GSK525768A ( GSK 525768A;GSK-525768A )

产品货号. M11076 CAS No. 1260530-25-3

GSK525768A is an enantiomer, negative control compound of I-BET762 (GSK525762A).

纯度: >98% (HPLC)

COA

Datasheet

HNMR

HPLC

MSDS

Handing Instructions

规格	价格/人民币	库存	数量
5MG	￥2811	有现货
50MG	￥12393	有现货
100MG	￥16119	有现货
200MG	获取报价	有现货
500MG	获取报价	有现货
1G	获取报价	有现货

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生物学信息

产品名称

GSK525768A
注意事项

本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
产品简述

GSK525768A is an enantiomer, negative control compound of I-BET762 (GSK525762A).
产品描述

GSK525768A is an enantiomer, negative control compound of I-BET762 (GSK525762A), shows no activity against BET family proteins BRD2, BRD3 and BRD4.
同义词

GSK 525768A;GSK-525768A
通路

Chromatin/Epigenetic
靶点

Bromodomain
受体

Bromodomain
研究领域

Inflammation/Immunology
适应症

——

化学信息

CAS Number

1260530-25-3
分子量

423.90
分子式

C22H22ClN5O2
纯度

>98% (HPLC)
溶解度

10 mM in DMSO
SMILES

CCNC(=O)CC1C2=NN=C(N2C3=C(C=C(C=C3)OC)C(=N1)C4=CC=C(C=C4)Cl)C
化学全称

4H-[1,2,4]Triazolo[4,3-a][1,4]benzodiazepine-4-acetamide, 6-(4-chlorophenyl)-N-ethyl-8-methoxy-1-methyl-, (4R)-

运输与储存

储存条件

(-20℃)
运输条件

With Ice Pack
稳定性

≥ 2 years

参考文献

1. Nicodeme E, et al. Nature. 2010 Dec 23;468(7327):1119-23.

计算器

浓度计算器

摩尔计算器

分子量计算器

产品手册

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