GSK269962A
CAS No. 850664-21-0
GSK269962A ( GSK 269962 )
产品货号. M17614 CAS No. 850664-21-0
GSK269962 is a selective ROCK(Rho-associated protein kinase) inhibitor with IC50 values of 1.6 and 4 nM for ROCK1 and ROCK2, respectively.
纯度: 98%
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
规格 | 价格/人民币 | 库存 | 数量 |
2MG | ¥421 | 有现货 |
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5MG | ¥664 | 有现货 |
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10MG | ¥1239 | 有现货 |
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25MG | ¥2616 | 有现货 |
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50MG | ¥3880 | 有现货 |
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100MG | ¥5573 | 有现货 |
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200MG | 获取报价 | 有现货 |
|
500MG | 获取报价 | 有现货 |
|
1G | 获取报价 | 有现货 |
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生物学信息
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产品名称GSK269962A
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注意事项本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
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产品简述GSK269962 is a selective ROCK(Rho-associated protein kinase) inhibitor with IC50 values of 1.6 and 4 nM for ROCK1 and ROCK2, respectively.
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产品描述GSK269962 is a selective ROCK(Rho-associated protein kinase) inhibitor with IC50 values of 1.6 and 4 nM for ROCK1 and ROCK2, respectively.
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同义词GSK 269962
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通路Angiogenesis
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靶点VEGFR
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受体MSK1; ROCK1; ROCK2; RSK1
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研究领域Cardiovascular Disease
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适应症——
化学信息
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CAS Number850664-21-0
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分子量570.61
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分子式C29H30N8O5
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纯度98%
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溶解度DMSO : ≥ 30 mg/mL; 52.58 mM
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SMILESCCn1c2cc(ncc2nc1c1nonc1N)Oc1cccc(c1)NC(=O)c1ccc(cc1)OCCN1CCOCC1
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化学全称——
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1. Doe C, et al. Novel Rho kinase inhibitors with anti-inflammatory and vasodilatory activities. J Pharmacol Exp Ther. 2007 Jan;320(1):89-98. Epub 2006 Oct 3.
产品手册
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