GSK-812 ( GSK812 )

产品货号. M15383 CAS No. 630407-66-8

COA

Datasheet

HNMR

HPLC

MSDS

Handing Instructions

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产品名称

GSK-812
注意事项

本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
产品简述

GSK-812 is a potent neuroprotectant that can induce GDNF in normal and diseased retina.
产品描述

GSK-812 is a potent neuroprotectant that can induce GDNF in normal and diseased retina, shows has polypharmacology antagonizing multiple receptors, including D2 and D3 receptors, and 5-HT2A, 2C, and 5-HT6 receptors.
同义词

GSK812
通路

Endocrinology/Hormones
靶点

5-HT Receptor
受体

5-HT Receptor
研究领域

——
适应症

——

CAS Number

630407-66-8
分子量

472.00
分子式

C25H26ClNO4S
纯度

>98% (HPLC)
溶解度

——
SMILES

CN1CCC2=CC(=C(C=C2CC1)S(=O)(=O)C3=CC=C(C=C3)OCC4=CC=C(C=C4)Cl)OC
化学全称

7-[4-(4-chloro-benzyloxy)-benzenesulfonyl]-8-methoxy-3-methyl-2,3,4,5-tetrahydro-1H-3-benzazepine

1. Baranov P, et al. J Ocul Pharmacol Ther. 2017 Jun;33(5):412-422.

计算器

产品手册

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