
Fezolamine
CAS No. 80410-36-2
Fezolamine ( —— )
产品货号. M36171 CAS No. 80410-36-2
Fezolamine is a novel orally available non-tricyclic compound with antidepressant activity. It is three to two times more selective in blocking synaptosomal uptake of [3H]norepinephrine than uptake of [4H]3-hydroxytryptamine or [3H]dopamine in vitro. It blocked the inhibitory effects of rifampicin and tetraphenyl in classical behavioral tests using monoamine-depleted animals.
纯度: >98% (HPLC)






规格 | 价格/人民币 | 库存 | 数量 |
2MG | ¥1447 | 有现货 |
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5MG | ¥2100 | 有现货 |
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10MG | ¥3149 | 有现货 |
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25MG | ¥5106 | 有现货 |
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50MG | ¥7257 | 有现货 |
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100MG | ¥9639 | 有现货 |
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500MG | ¥19355 | 有现货 |
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1G | 获取报价 | 有现货 |
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生物学信息
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产品名称Fezolamine
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注意事项本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
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产品简述Fezolamine is a novel orally available non-tricyclic compound with antidepressant activity. It is three to two times more selective in blocking synaptosomal uptake of [3H]norepinephrine than uptake of [4H]3-hydroxytryptamine or [3H]dopamine in vitro. It blocked the inhibitory effects of rifampicin and tetraphenyl in classical behavioral tests using monoamine-depleted animals.
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产品描述Fezolamine is a novel orally available non-tricyclic compound with antidepressant activity. It is three to two times more selective in blocking synaptosomal uptake of [3H]norepinephrine than uptake of [4H]3-hydroxytryptamine or [3H]dopamine in vitro. It blocked the inhibitory effects of rifampicin and tetraphenyl in classical behavioral tests using monoamine-depleted animals.
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体外实验——
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体内实验——
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同义词——
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通路Neuroscience
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靶点Norepinephrine
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受体Norepinephrine
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研究领域——
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适应症——
化学信息
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CAS Number80410-36-2
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分子量305.42
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分子式C20H23N3
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纯度>98% (HPLC)
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溶解度——
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SMILESC(CCN(C)C)N1C=C(C(=N1)C2=CC=CC=C2)C3=CC=CC=C3
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化学全称——
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
产品手册




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Fezolamine
Fezolamine is a novel orally available non-tricyclic compound with antidepressant activity. It is three to two times more selective in blocking synaptosomal uptake of [3H]norepinephrine than uptake of [4H]3-hydroxytryptamine or [3H]dopamine in vitro. It blocked the inhibitory effects of rifampicin and tetraphenyl in classical behavioral tests using monoamine-depleted animals.