Cisapride ( Kaudalit; Kinestase; Prepulsid; Presid; Pridesia; Propulsid )

产品货号. M16029 CAS No. 81098-60-4

COA

Datasheet

HNMR

HPLC

MSDS

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产品名称

Cisapride
注意事项

本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
产品简述

Cisapride is a gastroprokinetic agent, a drug that increases motility in the upper gastrointestinal tract.
产品描述

Cisapride is a gastroprokinetic agent, a drug that increases motility in the upper gastrointestinal tract. It acts directly as a serotonin 5-HT4 receptor agonist and indirectly as a parasympathomimetic. Stimulation of the serotonin receptors increases acetylcholine release in the enteric nervous system.
同义词

Kaudalit; Kinestase; Prepulsid; Presid; Pridesia; Propulsid
通路

Endocrinology/Hormones
靶点

5-HT Receptor
受体

5-HT; Potassium Channel
研究领域

Neurological Disease
适应症

——

CAS Number

81098-60-4
分子量

465.95
分子式

C23H29ClFN3O4
纯度

>98%(HPLC)
溶解度

Water: 2.71 mg/L
SMILES

O=C(N[C@H]1[C@@H](OC)CN(CCCOC2=CC=C(F)C=C2)CC1)C3=CC(Cl)=C(N)C=C3OC
化学全称

Benzamide, 4-amino-5-chloro-N-(1-(3-(4-fluorophenoxy)propyl)-3-methoxy-4-piperidinyl)-2-methoxy-, cis-

1.Nagakura Y, et al. Pharmacol Res. 1999 May;39(5):375-82.

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