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Amperozide
CAS No. 75558-90-6
Amperozide ( FG 5606 | Amperozida | Amperozidum )
产品货号. M27751 CAS No. 75558-90-6
Amperozide 是一种 5-HT2 拮抗剂。
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| 规格 | 价格/人民币 | 库存 | 数量 |
| 5MG | ￥2722 | 有现货 |
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| 10MG | ￥4026 | 有现货 |
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| 25MG | ￥6423 | 有现货 |
|
| 50MG | ￥9153 | 有现货 |
|
| 100MG | ￥12312 | 有现货 |
|
| 200MG | 获取报价 | 有现货 |
|
| 500MG | 获取报价 | 有现货 |
|
| 1G | 获取报价 | 有现货 |
|
生物学信息
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产品名称Amperozide
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注意事项本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
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产品简述Amperozide 是一种 5-HT2 拮抗剂。
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产品描述Amperozide, a 5-HT2 antagonist, attenuates craving for cocaine by rats and reduces agonistic behaviors such as slashing and biting in pigs.(In Vitro):Amperozide inhibited the amphetamine-stimulated release of dopamine from perfused rat striatal tissue in a dose-dependent manner. With 1 and 10 microM amperozide there was significant inhibition of the amphetamine-stimulated release of dopamine, to 44 and 36% of control. In contrast, 10 microM amperozide significantly strengthened the electrically stimulated release of dopamine from perfused striatal slices. Amperozide 1-10 microM had no significant effect on the potassium-stimulated release of dopamine. 10 microM amperozide also slightly increased the basal release of 3H-dopamine from perfused striatal tissue.
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体外实验——
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体内实验——
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同义词FG 5606 | Amperozida | Amperozidum
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通路Endocrinology/Hormones
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靶点5-HT Receptor
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受体——
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研究领域——
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适应症——
化学信息
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CAS Number75558-90-6
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分子量401.5
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分子式C23H29F2N3O
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纯度>98% (HPLC)
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溶解度——
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SMILESO=C(N1CCN(CCCC(C2=CC=C(F)C=C2)C3=CC=C(F)C=C3)CC1)NCC
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化学全称——
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1.Morse MA, et al. Structure-activity relationships for inhibition of 4-(methylnitrosamino)-1-(3-pyridyl)-1-butanone lung tumorigenesis by arylalkyl isothiocyanates in A/J mice. Cancer Res. 1991;51(7):1846-1850.
产品手册
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