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CMP8
CAS No. 851107-28-3
CMP8 ( —— )
产品货号. M26655 CAS No. 851107-28-3
CMP8 is a selective ligand for estrogen receptor. CMP8 binds to the mutant estrogen receptor ligand binding domain (ERLBD).
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| 规格 | 价格/人民币 | 库存 | 数量 |
| 5MG | ￥4212 | 有现货 |
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| 10MG | ￥6018 | 有现货 |
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| 25MG | ￥9315 | 有现货 |
|
| 50MG | ￥12555 | 有现货 |
|
| 100MG | ￥16038 | 有现货 |
|
| 200MG | 获取报价 | 有现货 |
|
| 500MG | 获取报价 | 有现货 |
|
| 1G | 获取报价 | 有现货 |
|
生物学信息
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产品名称CMP8
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注意事项本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
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产品简述CMP8 is a selective ligand for estrogen receptor. CMP8 binds to the mutant estrogen receptor ligand binding domain (ERLBD).
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产品描述CMP8 is a selective ligand for estrogen receptor. CMP8 binds to the mutant estrogen receptor ligand binding domain (ERLBD). CMP8 has IC50 values of 29 nM , 41 nM, 1100 nM and 2200 nM for MGERα, MGRERα, hERα and hERβ, respectively.(In Vivo):CMP8 is dosed in male Balb-c mice (4 mg/kg, ip). In mammalian cells, the plasma concentration after 4 h is 1.5-fold its EC50. It has a Cmax of 0.5 μM after 30 min.
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同义词——
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通路Endocrinology/Hormones
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靶点Estrogen Receptor/ERR
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受体——
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研究领域——
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适应症——
化学信息
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CAS Number851107-28-3
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分子量528.1
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分子式C33H34ClNO3
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纯度>98% (HPLC)
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溶解度——
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SMILESOc1ccc2C3=C(C(=O)CCC3(Cc3ccc(Cl)cc3)Cc2c1)c1ccc(OCCN2CCCCC2)cc1
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化学全称——
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1.Wu WN, et al. Biotransformation of an antihypertensive arylalkylamine analogue in the rat. Xenobiotica. 1998 Oct;28(10):957-72.
产品手册
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