Valspodar ( PSC-833;SDZ PSC-833 )

产品货号. M10809 CAS No. 121584-18-7

A highly potent multidrug-resistance modifier that acts as a P-glycoprotein inhibitor.

纯度: >98% (HPLC)

COA

Datasheet

HNMR

HPLC

MSDS

Handing Instructions

规格	价格/人民币	库存	数量
10MG	￥12069	有现货
100MG	获取报价	有现货
200MG	获取报价	有现货
500MG	获取报价	有现货
1G	获取报价	有现货

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生物学信息

产品名称

Valspodar
注意事项

本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
产品简述

A highly potent multidrug-resistance modifier that acts as a P-glycoprotein inhibitor.
产品描述

A highly potent multidrug-resistance modifier that acts as a P-glycoprotein inhibitor; exhibits effectivity at preventing cancer cell resistance to chemotherapeutics.Blood Cancer Phase 2 Discontinued
同义词

PSC-833;SDZ PSC-833
通路

Membrane Transporter/Ion Channel
靶点

P-glycoprotein
受体

P-glycoprotein
研究领域

Cancer
适应症

Blood cancer

化学信息

CAS Number

121584-18-7
分子量

1214.62
分子式

C63H111N11O12
纯度

>98% (HPLC)
溶解度

DMSO: 12 mg/mL
SMILES

O=C([C@H](C(C)C)N(C)C([C@H](CC(C)C)N(C)C([C@H](CC(C)C)N(C)C([C@@H](C)NC([C@H](C)NC([C@H](CC(C)C)N(C)C([C@H](C(C)C)NC([C@H](CC(C)C)N(C)C(CN(C)C([C@H](C(C)C)N1)=O)=O)=O)=O)=O)=O)=O)=O)=O)N(C)[C@@H](C([C@H](C)C/C=C/C)=O)C1=O
化学全称

Cyclosporin A, 6-[(2S,4R,6E)-4-methyl-2-(methylamino)-3-oxo-6-octenoic acid]-7-L-valine-

运输与储存

储存条件

(-20℃)
运输条件

With Ice Pack
稳定性

≥ 2 years

参考文献

1. Boesch D, et al. Cancer Res. 1991 Aug 15;51(16):4226-33.
2. Ehrlich PH, et al. Anticancer Res. 1997 Jan-Feb;17(1A):129-33.
3. Hu XF, et al. Clin Cancer Res. 1996 Apr;2(4):713-20.

计算器

浓度计算器

摩尔计算器

分子量计算器

产品手册

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