UF-010
CAS No. 537672-41-6
UF-010 ( UF010;UF 010 )
产品货号. M14914 CAS No. 537672-41-6
A potent and selective inhibitor of class I HDACs.
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
规格 | 价格/人民币 | 库存 | 数量 |
10MG | ¥373 | 有现货 |
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25MG | ¥689 | 有现货 |
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50MG | ¥1199 | 有现货 |
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100MG | ¥2001 | 有现货 |
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200MG | ¥2600 | 有现货 |
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500MG | 获取报价 | 有现货 |
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1G | 获取报价 | 有现货 |
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生物学信息
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产品名称UF-010
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注意事项本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
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产品简述A potent and selective inhibitor of class I HDACs.
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产品描述A potent and selective inhibitor of class I HDACs with IC50s of 0.5/0.1/0.06/1.5/9.1/15.3/44.5 uM for HDAC1/2/3/8/6/10/11 respectively; shows no effect on HDAC4/5/7/9(>100 uM); induces the accumulation of protein acetylation and inhibits proliferation of NCI-60 panel of cancer cell lines (mean GI50=2.94 uM); a competitive with a fast-on/slow-off HDAC-binding mechanism.
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同义词UF010;UF 010
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通路Cell Cycle/DNA Damage
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靶点HDAC
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受体HDAC
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研究领域Cancer
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适应症——
化学信息
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CAS Number537672-41-6
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分子量271.15
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分子式C11H15BrN2O
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纯度>98% (HPLC)
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溶解度10 mM in DMSO
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SMILESO=C(NNCCCC)C1=CC=C(Br)C=C1
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化学全称Benzoic acid, 4-bromo-, 2-butylhydrazide
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1. Wang Y, et al. Chem Biol. 2015 Feb 19;22(2):273-84.
产品手册
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