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Tetomilast
CAS No. 145739-56-6
Tetomilast ( OPC-6535 )
产品货号. M11976 CAS No. 145739-56-6
Tetomilast (OPC-6535) is a superoxide anion production inhibitor that inhibits PDE4 and proinflammatory functions.
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| 规格 | 价格/人民币 | 库存 | 数量 |
| 5MG | ￥7857 | 有现货 |
|
| 100MG | 获取报价 | 有现货 |
|
| 200MG | 获取报价 | 有现货 |
|
| 500MG | 获取报价 | 有现货 |
|
| 1G | 获取报价 | 有现货 |
|
生物学信息
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产品名称Tetomilast
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注意事项本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
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产品简述Tetomilast (OPC-6535) is a superoxide anion production inhibitor that inhibits PDE4 and proinflammatory functions.
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产品描述Tetomilast (OPC-6535) is a superoxide anion production inhibitor that inhibits PDE4 and proinflammatory functions of leukocytes including superoxide production and cytokine release; attenuates sepsis-induced acute lung injury.COPD Phase 2 Clinical
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同义词OPC-6535
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通路Angiogenesis
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靶点PDE
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受体PDE
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研究领域Inflammation/Immunology
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适应症COPD
化学信息
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CAS Number145739-56-6
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分子量370.42
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分子式C19H18N2O4S
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纯度>98% (HPLC)
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溶解度——
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SMILESO=C(C1=NC(C2=CSC(C3=CC=C(OCC)C(OCC)=C3)=N2)=CC=C1)O
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化学全称6-[2-(3,4-diethoxyphenyl)-1,3-thiazol-4-yl]pyridine-2-carboxylic acid
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1. Schreiber S, et al. Gastroenterology. 2007 Jan;132(1):76-86.
2. Bloomfield GL, et al. J Surg Res. 1997 Sep;72(1):70-7.
3. Ejiri S, et al. Transplant Proc. 2000 Mar;32(2):318-21.
2. Bloomfield GL, et al. J Surg Res. 1997 Sep;72(1):70-7.
3. Ejiri S, et al. Transplant Proc. 2000 Mar;32(2):318-21.
产品手册
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