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Difamilast

CAS No. 937782-05-3

Difamilast ( OPA-15406;OPA15406 )

产品货号. M16718 CAS No. 937782-05-3

Difamilast (OPA-15406) is a novel potent, selective phosphodiesterase IV (PDE4) inhibitor with preference for PDE4B (IC50=11.2 nM).

纯度: >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
规格 价格/人民币 库存 数量
5MG ¥2657 有现货
10MG ¥4277 有现货
25MG ¥6958 有现货
50MG ¥9639 有现货
100MG ¥12798 有现货
200MG 获取报价 有现货
500MG 获取报价 有现货
1G 获取报价 有现货

生物学信息

  • 产品名称
    Difamilast
  • 注意事项
    本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
  • 产品简述
    Difamilast (OPA-15406) is a novel potent, selective phosphodiesterase IV (PDE4) inhibitor with preference for PDE4B (IC50=11.2 nM).
  • 产品描述
    Difamilast (OPA-15406) is a novel potent, selective phosphodiesterase IV (PDE4) inhibitor with preference for PDE4B (IC50=11.2 nM).Dermatitis Phase 2 Clinical
  • 同义词
    OPA-15406;OPA15406
  • 通路
    Angiogenesis
  • 靶点
    PDE
  • 受体
    PDE
  • 研究领域
    Inflammation/Immunology
  • 适应症
    Dermatitis

化学信息

  • CAS Number
    937782-05-3
  • 分子量
    446.45
  • 分子式
    3H24F2N2O5
  • 纯度
    >98% (HPLC)
  • 溶解度
    ——
  • SMILES
    O=C(NCC1=COC(C2=CC=C(OC(F)F)C(OC(C)C)=C2)=N1)C3=CC=CC=C3OCC
  • 化学全称
    N-({2-[4-(difluoromethoxy)-3-(propan-2-yloxy)phenyl]-1,3-oxazol-4-yl}methyl)-2-ethoxybenzamide

运输与储存

  • 储存条件
    (-20℃)
  • 运输条件
    With Ice Pack
  • 稳定性
    ≥ 2 years

参考文献

1.Hanifin JM, et al. J Am Acad Dermatol. 2016 Aug;75(2):297-305.
产品手册
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