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Talnetant
CAS No. 174636-32-9
Talnetant ( SB 223412 )
产品货号. M20780 CAS No. 174636-32-9
Talnetant is a selective competitive brain-penetrant NK3 receptor antagonist with the ability to modulate mesolimbic and mesocortical dopaminergic neurotransmission.
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| 规格 | 价格/人民币 | 库存 | 数量 |
| 2MG | ￥413 | 有现货 |
|
| 5MG | ￥680 | 有现货 |
|
| 10MG | ￥1069 | 有现货 |
|
| 25MG | ￥2260 | 有现货 |
|
| 50MG | ￥4172 | 有现货 |
|
| 100MG | ￥6342 | 有现货 |
|
| 200MG | 获取报价 | 有现货 |
|
| 500MG | 获取报价 | 有现货 |
|
| 1G | 获取报价 | 有现货 |
|
生物学信息
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产品名称Talnetant
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注意事项本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
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产品简述Talnetant is a selective competitive brain-penetrant NK3 receptor antagonist with the ability to modulate mesolimbic and mesocortical dopaminergic neurotransmission.
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产品描述Talnetant is a selective competitive brain-penetrant NK3 receptor antagonist with the ability to modulate mesolimbic and mesocortical dopaminergic neurotransmission.
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同义词SB 223412
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通路GPCR/G Protein
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靶点Neurokinin Receptor
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受体NK3
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研究领域Metabolic Disease
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适应症Chronic obstructive pulmonary disease; Cough; Irritable bowel syndrome
化学信息
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CAS Number174636-32-9
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分子量382.45
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分子式C25H22N2O2
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纯度>98% (HPLC)
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溶解度DMSO:100 mg/mL (261.47 mM)
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SMILESCCC(NC(=O)c1c(O)c(-c2ccccc2)nc2ccccc12)c1ccccc1
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化学全称3-hydroxy-2-phenyl-N-[(1S)-1-phenylpropyl]quinoline-4-carboxamide
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1.Dawson L A Cato K J Scott C et al. In Vitro and In Vivo Characterization of the Non-peptide NK3 Receptor Antagonist SB-223412 (Talnetant): Potential Therapeutic Utility in the Treatment of Schizophrenia[J]. Neuropsychopharmacology 2008 33(7):1642-1652.
产品手册
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