Talampanel ( GYKI-53773; LY-300164 )

产品货号. M26835 CAS No. 161832-65-1

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产品名称

Talampanel
注意事项

本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
产品简述

Talampanel is an orally and selective α-amino-3-hydroxy-5-methyl-4-isoxazolepropionate receptor antagonist with anti-seizure activity.
产品描述

Talampanel is an orally and selective α-amino-3-hydroxy-5-methyl-4-isoxazolepropionate receptor antagonist with anti-seizure activity. Talampanel (IVAX) has neuroprotective effects in rodent stroke models.(In Vivo):Talampanel (p.o.; 5 mg/kg; once a day; 2 weeks) decreases motoneuronal calcium in a mouse model of ALS .
同义词

GYKI-53773; LY-300164
通路

Apoptosis
靶点

Apoptosis
受体

ASK1
研究领域

——
适应症

——

1.Kawarazaki Y, Ichijo H, Naguro I. Apoptosis signal-regulating kinase 1 as a therapeutic target. Expert Opin Ther Targets. 2014 Jun;18(6):651-64.

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