Tadalafil
CAS No. 171596-29-5
Tadalafil ( IC351, IC-351, IC 351, Tadalafil, Adcirca, Cialis )
产品货号. M12614 CAS No. 171596-29-5
Tadalafil is a potent phosphodiesterase-5 (PDE5) inhibitor (IC50=1 nM).
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
规格 | 价格/人民币 | 库存 | 数量 |
25MG | ¥405 | 有现货 |
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50MG | ¥591 | 有现货 |
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100MG | ¥907 | 有现货 |
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200MG | ¥1523 | 有现货 |
|
500MG | 获取报价 | 有现货 |
|
1G | 获取报价 | 有现货 |
|
生物学信息
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产品名称Tadalafil
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注意事项本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
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产品简述Tadalafil is a potent phosphodiesterase-5 (PDE5) inhibitor (IC50=1 nM).
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产品描述Tadalafil is a potent phosphodiesterase-5 (PDE5) inhibitor (IC50=1 nM); no inhibition on most of the other families of PDEs, with the exception of PDE11.Sexual Dysfunction Approved
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同义词IC351, IC-351, IC 351, Tadalafil, Adcirca, Cialis
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通路Angiogenesis
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靶点PDE
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受体PDE5
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研究领域Endocrinology
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适应症Sexual Dysfunction
化学信息
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CAS Number171596-29-5
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分子量389.40
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分子式C22H19N3O4
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纯度>98% (HPLC)
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溶解度DMSO: ≥ 52 mg/mL
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SMILESO=C([C@@]1([H])CC2=C([C@@H](C3=CC(OCO4)=C4C=C3)N15)NC6=C2C=CC=C6)N(C)CC5=O
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化学全称Pyrazino[1',2':1,6]pyrido[3,4-b]indole-1,4-dione, 6-(1,3-benzodioxol-5-yl)-2,3,6,7,12,12a-hexahydro-2-methyl-, (6R,12aR)-
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1. Blount MA, et al. Mol Pharmacol, 2004, 66(1), 144-152.
2. Ring BJ, et al. Clin Pharmacol Ther, 2005, 77(1), 63-75.
2. Ring BJ, et al. Clin Pharmacol Ther, 2005, 77(1), 63-75.
产品手册
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