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SIS17

CAS No. 2374313-54-7

SIS17 ( —— )

产品货号. M20333 CAS No. 2374313-54-7

SIS17 is a potent and selective HDAC 11 inhibitor with an IC50 value of 0.83 μM. SIS17 is active in cells and inhibited the demyristoylation of a known HDAC11 substrate serine hydroxymethyl transferase 2 without inhibiting other HDACs.

纯度: >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
规格 价格/人民币 库存 数量
5MG ¥478 有现货
10MG ¥794 有现货
25MG ¥1531 有现货
50MG ¥2608 有现货
100MG ¥4155 有现货
200MG 获取报价 有现货
500MG 获取报价 有现货
1G 获取报价 有现货

生物学信息

  • 产品名称
    SIS17
  • 注意事项
    本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
  • 产品简述
    SIS17 is a potent and selective HDAC 11 inhibitor with an IC50 value of 0.83 μM. SIS17 is active in cells and inhibited the demyristoylation of a known HDAC11 substrate serine hydroxymethyl transferase 2 without inhibiting other HDACs.
  • 产品描述
    SIS17 is a potent and selective HDAC 11 inhibitor with an IC50 value of 0.83 μM. SIS17 is active in cells and inhibited the demyristoylation of a known HDAC11 substrate serine hydroxymethyl transferase 2 without inhibiting other HDACs.
  • 同义词
    ——
  • 通路
    Cell Cycle/DNA Damage
  • 靶点
    HDAC
  • 受体
    HDAC11
  • 研究领域
    ——
  • 适应症
    ——

化学信息

  • CAS Number
    2374313-54-7
  • 分子量
    366.6
  • 分子式
    C21H38N2OS?
  • 纯度
    >98% (HPLC)
  • 溶解度
    DMSO:125 mg/mL?(340.97 mM)
  • SMILES
    CCCCCCCCCCCCCCCCNNC(=O)c1cccs1
  • 化学全称
    ——

运输与储存

  • 储存条件
    (-20℃)
  • 运输条件
    With Ice Pack
  • 稳定性
    ≥ 2 years

参考文献

1.Son S I Cao J Zhu C L et al. Activity-Guided Design of HDAC11-Specific Inhibitors[J]. ACS Chemical Biology 2019 14(7):1393-1397.
产品手册
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