SIS17
CAS No. 2374313-54-7
SIS17 ( —— )
产品货号. M20333 CAS No. 2374313-54-7
SIS17 is a potent and selective HDAC 11 inhibitor with an IC50 value of 0.83 μM. SIS17 is active in cells and inhibited the demyristoylation of a known HDAC11 substrate serine hydroxymethyl transferase 2 without inhibiting other HDACs.
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
规格 | 价格/人民币 | 库存 | 数量 |
5MG | ¥478 | 有现货 |
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10MG | ¥794 | 有现货 |
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25MG | ¥1531 | 有现货 |
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50MG | ¥2608 | 有现货 |
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100MG | ¥4155 | 有现货 |
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200MG | 获取报价 | 有现货 |
|
500MG | 获取报价 | 有现货 |
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1G | 获取报价 | 有现货 |
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生物学信息
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产品名称SIS17
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注意事项本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
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产品简述SIS17 is a potent and selective HDAC 11 inhibitor with an IC50 value of 0.83 μM. SIS17 is active in cells and inhibited the demyristoylation of a known HDAC11 substrate serine hydroxymethyl transferase 2 without inhibiting other HDACs.
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产品描述SIS17 is a potent and selective HDAC 11 inhibitor with an IC50 value of 0.83 μM. SIS17 is active in cells and inhibited the demyristoylation of a known HDAC11 substrate serine hydroxymethyl transferase 2 without inhibiting other HDACs.
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同义词——
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通路Cell Cycle/DNA Damage
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靶点HDAC
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受体HDAC11
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研究领域——
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适应症——
化学信息
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CAS Number2374313-54-7
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分子量366.6
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分子式C21H38N2OS?
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纯度>98% (HPLC)
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溶解度DMSO:125 mg/mL?(340.97 mM)
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SMILESCCCCCCCCCCCCCCCCNNC(=O)c1cccs1
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化学全称——
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1.Son S I Cao J Zhu C L et al. Activity-Guided Design of HDAC11-Specific Inhibitors[J]. ACS Chemical Biology 2019 14(7):1393-1397.
产品手册
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