SB-222200
CAS No. 174635-69-9
SB-222200 ( —— )
产品货号. M23788 CAS No. 174635-69-9
SB-222200 is a selective, reversible, and competitive antagonist of the human NK-3 receptor(Ki=4.4 nM).
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
规格 | 价格/人民币 | 库存 | 数量 |
5MG | ¥551 | 有现货 |
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10MG | ¥834 | 有现货 |
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25MG | ¥2049 | 有现货 |
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50MG | ¥3929 | 有现货 |
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100MG | ¥5613 | 有现货 |
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200MG | 获取报价 | 有现货 |
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500MG | 获取报价 | 有现货 |
|
1G | 获取报价 | 有现货 |
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生物学信息
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产品名称SB-222200
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注意事项本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
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产品简述SB-222200 is a selective, reversible, and competitive antagonist of the human NK-3 receptor(Ki=4.4 nM).
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产品描述SB-222200 is a selective, reversible, and competitive antagonist of the human NK-3 receptor(Ki=4.4 nM).
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同义词——
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通路GPCR/G Protein
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靶点Neurokinin Receptor
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受体NK3
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研究领域——
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适应症——
化学信息
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CAS Number174635-69-9
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分子量380.5
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分子式C26H24N2O
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纯度>98% (HPLC)
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溶解度DMSO:100 mg/mL (262.83 mM)
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SMILESO=C(C1=C(C)C(C2=CC=CC=C2)=NC3=CC=CC=C13)N[C@H](C4=CC=CC=C4)CC
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化学全称——
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1.Sarau HM, et al. Nonpeptide tachykinin receptor antagonists. II. Pharmacological and pharmacokinetic profile of SB-222200, a central nervous system penetrant, potent and selective NK-3 receptor antagonist. J Pharmacol Exp Ther. 2000 Oct;295(1):373-81.
产品手册
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