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Maropitant
CAS No. 147116-67-4
Maropitant ( —— )
产品货号. M20648 CAS No. 147116-67-4
Maropitant 是一种选择性神经激肽 (NK1) 受体拮抗剂。
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| 规格 | 价格/人民币 | 库存 | 数量 |
| 2MG | ￥348 | 有现货 |
|
| 5MG | ￥583 | 有现货 |
|
| 10MG | ￥988 | 有现货 |
|
| 25MG | ￥1596 | 有现货 |
|
| 50MG | ￥3013 | 有现货 |
|
| 100MG | ￥4504 | 有现货 |
|
| 500MG | ￥9882 | 有现货 |
|
| 1G | 获取报价 | 有现货 |
|
生物学信息
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产品名称Maropitant
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注意事项本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
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产品简述Maropitant 是一种选择性神经激肽 (NK1) 受体拮抗剂。
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产品描述Maropitant is a selective neurokinin (NK1) receptor antagonist.
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体外实验——
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体内实验Treatment with 1 mg/kg Maropitant citrate, significantly reduces the size of ulcerative dermatitis (UD) lesions in mice. Intravenous Maropitant decreases MAC by 16%. In contrast, epidural administration of either saline or Maropitant does not change the MAC (2.17% and 1.92 %, respectively).
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同义词——
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通路GPCR/G Protein
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靶点Neurokinin Receptor
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受体NK1
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研究领域——
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适应症——
化学信息
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CAS Number147116-67-4
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分子量468.67
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分子式C32H40N2O
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纯度>98% (HPLC)
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溶解度DMSO:33.33 mg/mL (71.12 mM)
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SMILESCOc1ccc(cc1CN[C@H]1C2CCN(CC2)[C@H]1C(c1ccccc1)c1ccccc1)C(C)(C)C
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化学全称——
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1.Hickman M A Cox S R Mahabir S et al. Safety pharmacokinetics and use of the novel NK‐1 receptor antagonist maropitant (Cerenia TM ) for the prevention of emesis and motion sickness in cats[J]. Journal of Veterinary Pharmacology and Therapeutics 2008 31(3):220-229.
产品手册
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