Revexepride ( SSP 002358;SPD-557 )

产品货号. M13507 CAS No. 219984-49-3

COA

Datasheet

HNMR

HPLC

MSDS

Handing Instructions

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产品名称

Revexepride
注意事项

本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
产品简述

Revexepride (SSP 002358;SPD-557) potent, highly selective 5-HT4 receptor agonist for the treatment of gastroesophageal reflux disease.
产品描述

Revexepride (SSP 002358;SPD-557) potent, highly selective 5-HT4 receptor agonist for the treatment of gastroesophageal reflux disease. Other Indication Phase 2 Discontinued
同义词

SSP 002358;SPD-557
通路

Endocrinology/Hormones
靶点

5-HT Receptor
受体

5-HT Receptor
研究领域

Other Indications
适应症

Other Disease

CAS Number

219984-49-3
分子量

425.95
分子式

C21H32ClN3O4
纯度

>98% (HPLC)
溶解度

——
SMILES

O=C(C1=CC(Cl)=C(N)C2=C1OC(C)(C)C2)NC[C@H]3[C@H](O)CN(CCCOC)CC3
化学全称

4-amino-5-chloro-N-(((3S,4S)-3-hydroxy-1-(3-methoxypropyl)piperidin-4-yl)methyl)-2,2-dimethyl-2,3-dihydrobenzofuran-7-carboxamide

1. Flach S, et al. Drug Des Devel Ther. 2016 Sep 27;10:3125-3132.
2. Shaheen NJ, et al. Aliment Pharmacol Ther. 2015 Apr;41(7):649-61.

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