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RK-287107
CAS No. 2171386-10-8
RK-287107 ( —— )
产品货号. M23984 CAS No. 2171386-10-8
RK-287107 is an effective and specific inhibitor of tankyrase (IC50s: 14.3 and 10.6 nM for tankyrase-1 and tankyrase-2, respectively).
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| 规格 | 价格/人民币 | 库存 | 数量 |
| 5MG | ￥1596 | 有现货 |
|
| 10MG | ￥2535 | 有现货 |
|
| 25MG | ￥4779 | 有现货 |
|
| 50MG | ￥6901 | 有现货 |
|
| 100MG | ￥9477 | 有现货 |
|
| 200MG | 获取报价 | 有现货 |
|
| 500MG | 获取报价 | 有现货 |
|
| 1G | 获取报价 | 有现货 |
|
生物学信息
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产品名称RK-287107
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注意事项本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
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产品简述RK-287107 is an effective and specific inhibitor of tankyrase (IC50s: 14.3 and 10.6 nM for tankyrase-1 and tankyrase-2, respectively).
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产品描述RK-287107 is an effective and specific inhibitor of tankyrase (IC50s: 14.3 and 10.6 nM for tankyrase-1 and tankyrase-2, respectively).
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同义词——
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通路Others
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靶点Other Targets
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受体tankyrase 1;tankyrase 2
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研究领域——
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适应症——
化学信息
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CAS Number2171386-10-8
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分子量416.5
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分子式C22H26F2N4O2
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纯度>98% (HPLC)
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溶解度DMSO:120 mg/mL (288.14 mM; Need ultrasonic)
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SMILESOCCN(C1)c2cc(F)cc(F)c2C1(CC1)CCN1C(N1)=NC(CCCC2)=C2C1=O
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化学全称——
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1.Mizutani A, et al. RK-287107, a potent and specific tankyrase inhibitor, blocks colorectal cancer cell growth in a preclinical model. Cancer Sci. 2018 Dec;109(12):4003-4014.
产品手册
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