PfDHODH-IN-2
CAS No. 425629-94-3
PfDHODH-IN-2 ( —— )
产品货号. M22750 CAS No. 425629-94-3
PfDHODH-IN-2 is a dihydrothiophenone derivative, is a potent Plasmodium falciparum dihydroorotate dehydrogenase (PfDHODH, IC50 : 1.11 μM) inhibitor.
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
规格 | 价格/人民币 | 库存 | 数量 |
5MG | ¥1320 | 有现货 |
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10MG | ¥2001 | 有现货 |
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25MG | ¥3686 | 有现货 |
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50MG | ¥5443 | 有现货 |
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100MG | ¥7744 | 有现货 |
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200MG | 获取报价 | 有现货 |
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500MG | 获取报价 | 有现货 |
|
1G | 获取报价 | 有现货 |
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生物学信息
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产品名称PfDHODH-IN-2
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注意事项本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
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产品简述PfDHODH-IN-2 is a dihydrothiophenone derivative, is a potent Plasmodium falciparum dihydroorotate dehydrogenase (PfDHODH, IC50 : 1.11 μM) inhibitor.
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产品描述PfDHODH-IN-2 is a dihydrothiophenone derivative, is a potent Plasmodium falciparum dihydroorotate dehydrogenase (PfDHODH, IC50 : 1.11 μM) inhibitor .?It is used an antimalarial agent and can be used for the research of malaria.
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同义词——
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通路Metabolic Enzyme/Protease
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靶点Dehydrogenase
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受体PfDHODH
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研究领域——
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适应症——
化学信息
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CAS Number425629-94-3
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分子量297.76
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分子式C13H12ClNO3S
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纯度>98% (HPLC)
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溶解度DMSO:12 mg/mL?(40.3 mM;?Need ultrasonic)
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SMILESCCOC(=O)C1=C(Nc2ccc(Cl)cc2)SCC1=O
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化学全称——
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1.Minghao Xu, et al. Novel selective and potent inhibitors of malaria parasite dihydroorotate dehydrogenase: discovery and optimization of dihydrothiophenone derivatives. J Med Chem. 2013 Oct 24;56(20):7911-24.
产品手册
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