PCI-34051
CAS No. 950762-95-5
PCI-34051 ( PCI34051; PCI 34051; PCI-34051 )
产品货号. M16799 CAS No. 950762-95-5
PCI-34051 is a potent and specific HDAC8 inhibitor with IC50 of 10 nM.
纯度: >98%(HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
规格 | 价格/人民币 | 库存 | 数量 |
5MG | ¥446 | 有现货 |
|
10MG | ¥786 | 有现货 |
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25MG | ¥1580 | 有现货 |
|
50MG | ¥3013 | 有现货 |
|
100MG | ¥4836 | 有现货 |
|
500MG | ¥10206 | 有现货 |
|
1G | 获取报价 | 有现货 |
|
生物学信息
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产品名称PCI-34051
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注意事项本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
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产品简述PCI-34051 is a potent and specific HDAC8 inhibitor with IC50 of 10 nM.
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产品描述PCI-34051 is a potent and specific HDAC8 inhibitor with IC50 of 10 nM. It has greater than 200-fold selectivity over HDAC1 and 6, more than 1000-fold selectivity over HDAC2, 3, and 10.
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同义词PCI34051; PCI 34051; PCI-34051
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通路Cell Cycle/DNA Damage
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靶点HDAC
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受体HDAC1; HDAC10; HDAC2; HDAC6; HDAC8
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研究领域Cancer
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适应症——
化学信息
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CAS Number950762-95-5
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分子量296.32
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分子式C17H16N2O3
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纯度>98%(HPLC)
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溶解度DMSO:59 mg/mL (199.1 mM); Ethanol:<1 mg/mL (<1 mM); Water:<1 mg/mL (<1 mM)
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SMILESO=C(C1=CC2=C(C=C1)C=CN2CC3=CC=C(OC)C=C3)NO
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化学全称N-hydroxy-1-(4-methoxybenzyl)-1H-indole-6-carboxamide
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1.Balasubramanian S, et al. Leukemia. 2008, 22(5), 1026-1034.
产品手册
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